IP Library Granted Patent US 10,125,106
Granted Patent B2
US 10,125,106 · App. 15/629,068 · Granted Nov 13, 2018

Contrast agents for myocardial perfusion imaging

Inventors: David S. Casebier (Carlisle, MA); Ajay Purohit (Sudbury, MA); Heike S. Radeke (South Grafton, MA)
Assignee: Lantheus Medical Imaging, Inc.
C07D237/16A61K49/00A61K49/0002A61K49/0052A61K49/10A61K49/22A61K51/04A61K51/0421A61K51/0453A61K51/0459C07B59/002
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Quick Facts
Patent No.
US 10,125,106
App. No.
15/629,068
Granted
Nov 13, 2018
Kind
B2
Abstract

The present disclosure is directed, in part, to compounds and methods for imaging myocardial perfusion, comprising administering to a patient a contrast agent which comprises a compound that binds MC-1, and an imaging moiety, and scanning the patient using diagnostic imaging.

Claims (12)

1. A compound having the structure:

2. A composition, comprising:

the compound of claim 1 and a solvent.

3. A compound having the structure:

4. A composition comprising:

the compound of claim 3 and a solvent.

5. A precursor compound to a 18 F labeled contrast agent of formula:

wherein the precursor compound has the formula:

and L G is a leaving group that can be replaced in an S N 2 displacement reaction to produce the 18 F labeled contrast agent.

6. The precursor compound of claim 5 , wherein the precursor compound is provided in a solution.

7. The precursor compound of claim 5 , wherein the precursor compound is provided as a solid preparation.

8. The precursor compound of claim 7 , wherein the solid preparation is a lyophilized solid.

Assignments (6)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Oct 6, 2017
From: CASEBIER, DAVID S.; ROBINSON, SIMON P.; PUROHIT, AJAY; RADEKE, HEIKE S.; AZURE, MICHAEL T.; DISCHINO, DOUGLAS D.
To: BRISTOL-MYERS SQUIBB COMPANY
Reel/Frame 043802/0820 →
NUNC PRO TUNC ASSIGNMENT Recorded Oct 6, 2017
From: BRISTOL-MYERS SQUIBB COMPANY
To: BRISTOL-MYERS SQUIBB PHARMA COMPANY
Reel/Frame 043802/0856 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Oct 6, 2017
From: CASEBIER, DAVID S.; ROBINSON, SIMON P.; PUROHIT, AJAY; RADEKE, HEIKE S.; AZURE, MICHAEL T.; DISCHINO, DOUGLAS D.
To: BRISTOL-MYERS SQUIBB PHARMA COMPANY
Reel/Frame 043802/0867 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Oct 6, 2017
From: BRISTOL-MYERS SQUIBB PHARMA COMPANY
To: ACP LANTERN ACQUISITION, INC.
Reel/Frame 044141/0545 →
MERGER Recorded Oct 6, 2017
From: ACP LANTERN ACQUISITION, INC.
To: BRISTOL-MYERS SQUIBB MEDICAL IMAGING, INC.
Reel/Frame 044144/0742 →
CHANGE OF NAME Recorded Oct 6, 2017
From: BRISTOL-MYERS SQUIBB MEDICAL IMAGING, INC.
To: LANTHEUS MEDICAL IMAGING, INC.
Reel/Frame 044144/0764 →
Continuity (6)
Continuation 14845320 · Sep 4, 2015
Continuation 13529756 · Jun 21, 2012
Continuation 12014161 · Jan 15, 2008
Division 11055498 · Feb 10, 2005
Provisional Application 60544861 · Feb 13, 2004
Related Publication 20180009763A1 · Jan 11, 2018
Cited By (1)
US 12,527,884