IP Library Granted Patent US 10,358,443
Granted Patent B2
US 10,358,443 · App. 15/666,503 · Granted Jul 23, 2019

Heteroaryl amides as inhibitors of protein aggregation

Inventors: Wolfgang Wrasidlo (San Diego, CA); Emily M. Stocking (Encinitas, CA)
Assignee: UCB Biopharma SPRL
C07D417/12C07D403/12C07D413/12C07D417/14
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Quick Facts
Patent No.
US 10,358,443
App. No.
15/666,503
Granted
Jul 23, 2019
Kind
B2
Abstract

The present invention relates to certain heteroaryl amide compounds, pharmaceutical compositions containing them, and methods of using them, including methods for preventing, reversing, slowing, or inhibiting protein aggregation, and methods of treating diseases that are associated with protein aggregation, including neurodegenerative diseases such as Parkinson's disease, Alzheimer's disease, Lewy body disease, Parkinson's disease with dementia, fronto-temporal dementia, Huntington's Disease, amyotrophic lateral sclerosis, and multiple system atrophy, and cancer and melanoma.

Claims (7)

1. A method of treating Parkinson's disease, comprising administering to a subject in need of such treatment an effective amount of a compound that is

or a pharmaceutically acceptable salt thereof.

2. The method of claim 1 , wherein the compound is:

or a pharmaceutically acceptable salt thereof.

3. The method of claim 1 . wherein the compound is:

or a pharmaceutically acceptable salt thereof.

4. The method of claim 1 , wherein Parkinson's disease is Parkinson's disease with dementia.

Assignments (3)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Feb 22, 2019
From: NEUROPORE THERAPIES, INC.
To: UCB BIOPHARMA SPRL
Reel/Frame 048416/0889 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Nov 21, 2018
From: WRASIDLO, WOLFGANG; STOCKING, EMILY M.
To: NEUROPORE THERAPIES, INC.
Reel/Frame 048149/0375 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Mar 8, 2018
From: NEUROPORE THERAPIES, INC.
To: UCB BIOPHARMA SPRL
Reel/Frame 045150/0153 →
Continuity (5)
Continuation 14983243 · Dec 29, 2015
Continuation PCTUS2015013263 · Jan 28, 2015
Provisional Application 62078895 · Nov 12, 2014
Provisional Application 61933246 · Jan 29, 2014
Related Publication 20180093979A1 · Apr 5, 2018
Cited By (1)
US 12,247,071