IP Library Granted Patent US 10,751,415
Granted Patent B2
US 10,751,415 · App. 15/680,187 · Granted Aug 25, 2020

Anti-TIGIT antibodies, anti-PVRIG antibodies and combinations thereof

Inventors: Mark White (Antioch, CA); Sandeep Kumar (San Bruno, CA); Christopher Chan (South San Francisco, CA); Spencer Liang (San Mateo, CA); Lance Stapleton (Oakland, CA); Andrew W. Drake (Mountain View, CA); Yosi Gozlan (Tel Aviv, IL); Ilan Vaknin (Tel Aviv, IL); Shirley Sameah-Greenwald (Kfar Saba, IL); Liat Dassa (Tel Aviv, IL); Zohar Tiran (Oranit, IL); Gad S. Cojocaru (Tel Aviv, IL); Maya Kotturi (Belmont, CA); Hsin-Yuan Cheng (San Mateo, CA); Kyle Hansen (San Francisco, CA); David Nisim Giladi (Netaniya, IL); Einav Safyon (Raanana, IL); Eran Ophir (Even Yehuda, IL); Leonard Presta (San Francisco, CA); Richard Theolis (Santa Cruz, CA); Radhika Desai (Brisbane, CA); Patrick Wall (Mill Valley, CA)
Assignee: Compugen Ltd.
A61K39/39558A61K39/39541A61P35/00C07K16/2803C07K16/2809C07K16/2818C07K16/2827A61K2039/505A61K2039/507A61K2039/572C07K2317/21C07K2317/24C07K2317/33C07K2317/34C07K2317/522C07K2317/524C07K2317/526C07K2317/53C07K2317/55C07K2317/56C07K2317/565C07K2317/622C07K2317/732C07K2317/76C07K2317/92C07K2317/94C07K2319/035C07K2319/33Y02A50/466
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Quick Facts
Patent No.
US 10,751,415
App. No.
15/680,187
Granted
Aug 25, 2020
Kind
B2
Abstract

Anti-PVRIG and anti-TIGIT antibodies are provided.

Claims (30)

1. A composition comprising an antigen binding domain that binds to human TIGIT (SEQ ID NO:97) comprising:

a) a variable heavy domain comprising SEQ ID NO:160; and

b) a variable light domain comprising SEQ ID NO:165.

2. A composition according to claim 1 wherein said composition is an antibody comprising:

a) a heavy chain comprising VH-CH1-hinge-CH2-CH3, wherein said VH comprises SEQ ID NO:160; and

b) a light chain comprising VL-VC, wherein said VL comprising SEQ ID NO:165 and VC is either kappa or lambda.

3. A composition according to claim 2 wherein the sequence said CH1-hinge-CH2-CH3 is selected from human IgG1, IgG2 and IgG4, and variants thereof.

4. A composition according to claim 2 wherein said heavy chain has SEQ ID NO:164 and said light chain has SEQ ID NO:169.

5. A composition according to claim 2 further comprising a second antibody that binds to a human checkpoint receptor protein.

6. A composition according to claim 5 wherein said second antibody binds human PD-1.

7. A composition according to claim 5 wherein said second antibody binds human PVRIG (SEQ ID NO:2).

8. A composition according to claim 7 wherein said second antibody comprises an antigen binding domain comprising a variable heavy domain comprising SEQ ID NO:5 and a variable light domain comprising SEQ ID NO:10.

9. A composition according to claim 7 wherein the heavy chain of said second antibody has SEQ ID NO:9 and the light chain of said second antibody has SEQ ID NO:14.

10. A composition according to claim 7 wherein said second antibody comprises an antigen binding domain comprising a variable heavy domain comprising SEQ ID NO:15 and a variable light domain comprising SEQ ID NO:20.

11. A composition according to claim 7 wherein the heavy chain of said second antibody has SEQ ID NO:19 and the light chain of said second antibody has SEQ ID NO:24.

12. A composition according to claim 7 wherein said second antibody comprises:

i) the vhCDR1, vhCDR2, and vhCDR3 from SEQ ID NO:5 and

ii) the v1CDR1, v1CDR2, and v1CDR3 from SEQ ID NO:10.

13. A composition comprising an antibody that binds to human TIGIT (SEQ ID NO:97) wherein said antibody comprises:

i) the vhCDR1, vhCDR2, and vhCDR3 from SEQ ID NO:160; and

ii) the v1CDR1, v1CDR2, and v1CDR3 from SEQ ID NO:165.

14. A composition according to claim 13 wherein said antibody comprises a CH1-hinge-CH2-CH3 region from human IgG1, IgG2, or IgG4, or variants thereof.

15. A composition according to claim 13 wherein said antibody comprises a VC region, wherein said VC is either kappa or lambda.

16. A composition according to claim 13 further comprising a second antibody that binds to a human checkpoint receptor protein.

17. A composition according to claim 16 wherein said second antibody binds human PD-1.

18. A composition according to claim 16 wherein said second antibody binds human PVRIG (SEQ ID NO:2).

19. A composition according to claim 18 wherein said second antibody comprises an antigen binding domain comprising a variable heavy domain comprising SEQ ID NO:5 and a variable light domain comprising SEQ ID NO:10.

20. A composition according to claim 18 wherein said second antibody comprises an antigen binding domain comprising a variable heavy domain comprising SEQ ID NO:15 and a variable light domain comprising SEQ ID NO:20.

21. A composition according to claim 18 wherein the heavy chain of said second antibody has SEQ ID NO:9 and the light chain of said second antibody has SEQ ID NO:14.

22. A composition according to claim 18 wherein the heavy chain of said second antibody has SEQ ID NO:19 and the light chain of said second antibody has SEQ ID NO:24.

Assignments (4)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Dec 18, 2017
From: WHITE, MARK; KUMAR, SANDEEP; CHAN, CHRISTOPHER; LIANG, SPENCER; STAPLETON, LANCE; DRAKE, ANDREW W.; KOTTURI, MAYA; CHENG, HSIN-YUAN; HANSEN, KYLE; THEOLIS, RICHARD; DESAI, RADHIKA; WALL, PATRICK
To: COMPUGEN USA, INC.
Reel/Frame 044426/0705 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Dec 18, 2017
From: PRESTA, LEONARD
To: COMPUGEN LTD.
Reel/Frame 044426/0730 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Dec 18, 2017
From: GOZLAN, YOSI; VAKNIN, ILAN; SAMEAH-GREENWALD, SHIRLEY; DASSA, LIAT; TIRAN, ZOHAR; COJOCARU, GAD S.; GILADI, DAVID NISIM; SAFYON, EINAV; OPHIR, ERAN
To: COMPUGEN LTD.
Reel/Frame 044426/0756 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Dec 18, 2017
From: COMPUGEN USA, INC.
To: COMPUGEN LTD.
Reel/Frame 044426/0777 →
Continuity (9)
Provisional Application 62376334 · Aug 17, 2016
Provisional Application 62513771 · Jun 1, 2017
Provisional Application 62376335 · Aug 17, 2016
Provisional Application 62417217 · Nov 3, 2016
Provisional Application 62513775 · Jun 1, 2017
Provisional Application 62477974 · Mar 28, 2017
Provisional Application 62513916 · Jun 1, 2017
Provisional Application 62538561 · Jul 28, 2017
Related Publication 20180305456A1 · Oct 25, 2018
Cited By (3)
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