IP Library Granted Patent US 12,178,846
Granted Patent B2
US 12,178,846 · App. 15/687,719 · Granted Dec 31, 2024

Methods of using gap junctions as therapeutic targets for the treatment of degenerative disorders of the retina

Inventor: Stewart Bloomfield (New York, NY)
Assignee: The Research Foundation for The State University of New York
A61K38/177A61K9/0019A61K9/0048A61K31/19A61K31/196A61K31/7105A61K38/16A61K45/06C12N15/1138C12N2310/11C12N2320/31
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Quick Facts
Patent No.
US 12,178,846
App. No.
15/687,719
Granted
Dec 31, 2024
Kind
B2
Abstract

The disclosure provides methods of treating a condition of the retina by administering an inhibitor of connexin 36 and/or an inhibitor of connexin 45 to a subject with a retinal condition. This disclosure further provides compositions for the treatment of a retinal condition which include an inhibitor of connexin 36 and/or an inhibitor of connexin 45.

Claims (3)

1. A method of treating glaucoma by blocking gap junctions comprising administering a therapeutically effective amount of a non-selective inhibitor of connexin 36 to a subject in need thereof, wherein said non-selective inhibitor is 18-Beta-glycyrrhetinic acid (18Beta-GA), and wherein the therapeutically effective amount is at a concentration of 25 μM.

2. The method of claim 1 , comprising repeat administration of said inhibitor for a period of 1 week to 1 year.

3. The method of claim 1 , wherein said administration is topical administration or intraocular injection.

Assignments (2)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Oct 4, 2024
From: BLOOMFIELD, STEWART
To: THE RESEARCH FOUNDATION FOR THE STATE UNIVERSITY OF NEW YORK
Reel/Frame 068801/0457 →
CONFIRMATORY LICENSE Recorded Jul 17, 2018
From: STATE UNIVERSITY NEW YORK
To: NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT
Reel/Frame 046364/0510 →
Continuity (3)
Division 15317171
Provisional Application 62011354 · Jun 12, 2014
Related Publication 20170354710A1 · Dec 14, 2017