IP Library Granted Patent US 10,562,901
Granted Patent B2
US 10,562,901 · App. 15/709,862 · Granted Feb 18, 2020

Temozolomide compounds, polymers prepared therefrom, and method of treating a disease

Inventors: Todd Emrick (South Deerfield, MA); Matthew Skinner (Amherst, MA); Sarah M. Ward (Amherst, MA); Banishree Saha (Greenfield, MA)
Assignee: THE UNIVERSITY OF MASSACHUSETTS
C07D487/04A61K31/787
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Quick Facts
Patent No.
US 10,562,901
App. No.
15/709,862
Granted
Feb 18, 2020
Kind
B2
Abstract

A temozolomide compound according to formula (I) is described, wherein R 1 , L 1 , and X are defined herein. The temozolomide compound can be used to prepare polymers comprising temozolomide. Additionally, the polymers comprising temozolomide can be particularly useful in the treatment of certain diseases.

Claims (18)

1. A temozolomide compound of structure (I)

wherein

X is —O— or —NH—;

n is 1;

L 1 is a divalent C 1-6 alkylene group; and

R 1 is a methacrylate group, a methacrylamide group, an acrylate group, or an acrylamide group.

2. A temozolomide compound of structure (I)

wherein

X is —O— or —NH—;

n is 1;

L 1 is a divalent di(C 2-6 alkylene) disulfide group; and

R 1 is a methacrylate group.

3. A temozolomide compound of structure (I)

wherein

X is —O— or —NH—;

n is 1;

L 1 is a divalent C 1-6 alkylene group; and

R 1 is a methacrylamide group.

Assignments (3)
CONFIRMATORY LICENSE Recorded Oct 4, 2021
From: UNIVERSITY OF MASSACHUSETTS AMHERST
To: NATIONAL SCIENCE FOUNDATION
Reel/Frame 057697/0743 →
CONFIRMATORY LICENSE Recorded Oct 1, 2019
From: UNIVERSITY OF MASSACHUSETTS, AMHERST
To: NATIONAL SCIENCE FOUNDATION
Reel/Frame 050584/0599 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Dec 8, 2017
From: EMRICK, TODD; SKINNER, MATTHEW; WARD, SARAH; SAHA, BANISHREE
To: THE UNIVERSITY OF MASSACHUSETTS
Reel/Frame 044336/0791 →
Continuity (2)
Provisional Application 62398078 · Sep 22, 2016
Related Publication 20180079754A1 · Mar 22, 2018