IP Library › Granted Patent US 10,214,548
Granted Patent B2
US 10,214,548 · App. 15/801,127 · Granted Feb 26, 2019

Boron containing small molecules as antiprotozoal agents

Inventors: Tsutomu Akama (Sunnyvale, CA); Eric Easom (Menlo Park, CA); Yvonne Freund (Los Altos, CA); Jacob J. Plattner (Berkeley, CA); Jessica Sligar (Cary, NC); Daitao Chen (Raleigh, NC); Jennifer Freeman (Durham, NC); Joe Perales (Durham, NC)
Assignee: Anacor Pharmaceuticals, Inc.
C07F5/025A61K31/69
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Quick Facts
Patent No.
US 10,214,548
App. No.
15/801,127
Granted
Feb 26, 2019
Kind
B2
Abstract

This invention provides, among other things, novel compounds useful for treating protozoal infections, pharmaceutical compositions containing such compounds, as well as combinations of these compounds with at least one additional therapeutically effective agent.

Claims (8)

1. A compound having a structure according to the following formulae:

wherein

R a is substituted or unsubstituted heteroaryl or substituted or unsubstituted heterocycloalkyl

or a salt thereof.

2. The compound of claim 1 , or a salt thereof, having a structure according to the following formulae:

3. The compound of claim 1 , or a salt thereof, having a structure according to the following formulae:

4. The compound of claim 1 , or a salt thereof, having a structure according to the following formulae:

5. The compound of claim 1 , or a salt thereof, which is:

Assignments (2)
CHANGE OF NAME Recorded Jan 11, 2024
From: ANACOR PHARMACEUTICALS, INC.
To: ANACOR PHARMACEUTICALS, LLC
Reel/Frame 066286/0038 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Nov 1, 2017
From: AKAMA, TSUTOMU; EASOM, ERIC; FREUND, YVONNE; PLATTNER, JACOB J.; SLIGAR, JESSICA; CHEN, DAITAO; FREEMAN, JENNIFER; PERALES, JOE
To: ANACOR PHARMACEUTICALS, INC.
Reel/Frame 044011/0851 →
Continuity (4)
Division 15439634 · Feb 22, 2017
Continuation 14765152
Provisional Application 61759981 · Feb 1, 2013
Related Publication 20180065994A1 · Mar 8, 2018