IP Library Granted Patent US 10,226,466
Granted Patent B2
US 10,226,466 · App. 15/836,482 · Granted Mar 12, 2019

Methods of treating fibrosis

Inventors: Toni Jauset González (Lleida, ES); Daniel Massó-Vallés (Barcelona, ES); Laura Soucek (Barcelona, ES)
Assignee: Pharmacyclics LLC
A61K31/519A61K31/7068C09B31/147
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Quick Facts
Patent No.
US 10,226,466
App. No.
15/836,482
Granted
Mar 12, 2019
Kind
B2
Abstract

Disclosed are methods of treating fibrosis in a patient, comprising administering to a patient in need thereof a therapeutically effective amount of an ACK inhibitor (e.g., a BTK inhibitor, such as for example an irreversible BTK inhibitor, such as for example, ibrutinib).

Claims (6)

1. A method of treating fibrosis, wherein the fibrosis is not associated with graft versus host disease (GVHD), comprising administering to a patient having fibrosis, wherein the fibrosis is not associated with GVHD, a therapeutically effective amount of a compound, which is 1-(R)-(3-(4-amino-3-(4-phenoxyphenyl)-1H-pyrazolo[3,4-d]pyrimidin-1-yl)piperidin-1-yl)prop-2-en-1-one (ibrutinib), of the structure:

thereby treating the fibrosis.

2. The method of claim 1 , wherein the fibrosis is of the liver, lung, kidney, bone marrow, heart, skin, intestine, or joints.

3. The method of claim 1 , wherein the fibrosis is of the liver.

4. The method of claim 1 , wherein the fibrosis is of the lung.

5. The method of claim 1 , wherein the patient has cirrhosis, or cystic fibrosis.

Assignments (2)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Dec 11, 2018
From: FUNDACIO PRIVADA INSTITUT D'INVESTIGACIO ONCOLOGICA DE VALL HEBRON
To: PHARMACYCLICS LLC
Reel/Frame 047742/0194 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Dec 11, 2018
From: GONZALEZ, TONI JAUSET; MASSÓ-VALLÉS, DANIEL; SOUCEK, LAURA
To: FUNDACIO PRIVADA INSTITUT D'INVESTIGACIO ONCOLOGICA DE VALL HEBRON
Reel/Frame 047786/0606 →
Continuity (3)
Division 14957294 · Dec 2, 2015
Provisional Application 62086945 · Dec 3, 2014
Related Publication 20180153896A1 · Jun 7, 2018
Cited By (1)
US 12,551,448