IP Library Granted Patent US 10,485,802
Granted Patent B2
US 10,485,802 · App. 15/897,138 · Granted Nov 26, 2019

Composition for inducing differentiation and protection of neural stem cells and method for inducing neuro-regeneration using the same composition

Inventors: Kang-Yell Choi (Seoul, KR); Mi-Yeon Kim (Seoul, KR); Sungho Han (Seoul, KR)
Assignee: GENUV Inc.
A61K31/519A61P25/16A61P25/28
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Quick Facts
Patent No.
US 10,485,802
App. No.
15/897,138
Granted
Nov 26, 2019
Kind
B2
Abstract

The present invention relates to a method of inducing neuro-regeneration comprising administering a MEK 1/2 inhibitor to a patient in need thereof. In the present invention, the MEK1/2 inhibitor induces neuro-regeneration by differentiating neural stem cells into neurons, by protecting neural stem cells and neurons against cytotoxicity of amyloid-betas, or by both of the above. Also, the present invention relates to a method of protecting neurons against neuronal loss or damage comprising administering a MEK1/2 inhibitor. In addition, this invention relates to a method of preventing or treating neurodegenerative disease due to neuronal loss or damage for patients in need thereof comprising administering a MEK 1/2 inhibitor.

Claims (11)

1. A method of treating Alzheimer's disease, comprising the step of administering trametinib to a patient diagnosed with Alzheimer's disease.

2. The method of claim 1 , wherein trametinib is administered in an amount sufficient to reduce a symptom associated with Alzheimer's disease.

3. The method of claim 1 , wherein trametinib is administered in an amount sufficient to induce neuro-regeneration.

4. The method of claim 3 , wherein the amount is sufficient to induce differentiation of a neural stem cell into a neuron in the patient.

5. The method of claim 4 , wherein the neuron differentiated from the neural stem cell is selected from the group consisting of: a dopaminergic neuron, a GABAergic neuron, a motor neuron, and a cholinergic neuron.

6. The method of claim 1 , wherein trametinib is administered in an amount sufficient to protect a neural stem cell or a neuron from cytotoxicity of amyloid-beta in the patient.

7. The method of claim 1 , wherein trametinib is administered in an amount of between 0.1 mg and 2 mg once daily.

8. The method of claim 7 , wherein trametinib is administered in an amount of not more than 1 mg once daily.

9. The method of claim 8 , wherein trametinib is administered in an amount of not more than 0.5 mg once daily.

10. The method of claim 1 , wherein trametinib is administered orally.

11. The method of claim 1 , wherein trametinib is administered orally in an amount of between 0.1 mg and 10 mg once daily.

Assignments (6)
CHANGE OF NAME Recorded Aug 15, 2019
From: SHINE BIOPHARMA, INC.
To: GENUV INC.
Reel/Frame 050074/0139 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Aug 6, 2019
From: KIM, MI-YEON
To: SHINE BIOHARMA, INC.
Reel/Frame 049981/0048 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Aug 6, 2019
From: HAN, SUNGHO
To: SHINE BIOPHARMA, INC.
Reel/Frame 049981/0052 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Aug 5, 2019
From: INDUSTRY-ACADEMIC COOPERATION FOUNDATION, YONSEI UNIVERSITY
To: SHINE BIOPHARMA, INC.
Reel/Frame 049962/0047 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Aug 1, 2019
From: CHOI, KANG-YELL
To: INDUSTRY-ACADEMIC COOPERATION FOUNDATION, YONSEI UNIVERSITY
Reel/Frame 049935/0710 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Aug 1, 2019
From: KIM, MI-YEON
To: INDUSTRY-ACADEMIC COOPERATION FOUNDATION, YONSEI UNIVERSITY
Reel/Frame 049937/0198 →
Priority Claims (2)
KR 10-2016-0158739 · Nov 25, 2016 · national
KR 10-2017-0036268 · Mar 22, 2017 · national
Continuity (2)
Continuation PCTKR2017013444 · Nov 23, 2017
Related Publication 20180169102A1 · Jun 21, 2018