IP Library › Granted Patent US 10,314,825
Granted Patent B2
US 10,314,825 · App. 15/903,279 · Granted Jun 11, 2019

Agent for treatment of PBC

Inventors: Mitsumasa Nakamura (Chuo-ku, JP); Satoshi Kojima (Chuo-ku, JP); Ryohei Tanigawa (Chuo-ku, JP)
Assignee: KOWA COMPANY, LTD.
A61K31/423A61K31/575A61P1/16
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Quick Facts
Patent No.
US 10,314,825
App. No.
15/903,279
Granted
Jun 11, 2019
Kind
B2
Abstract

The present invention relates to a pharmaceutical composition for the treatment of primary biliary cirrhosis (PBC), in which containing a therapeutically effective amount of (R)-2-[3-[[N-(benzoxazol-2-yl)-N-3-(4-methoxyphenoxy)propyl]aminomethyl]phenoxy] butyric acid, a salt thereof, or a solvate thereof.

Claims (5)

1. A method for the treatment of primary biliary cirrhosis, comprising administering (R)-2-[3-[[N-(benzoxazole-2-yl)-N-3-(4-methoxyphenoxy)propyl]aminomethyl]phenoxy] butyric acid, a salt thereof, or a solvate thereof to a patient in need thereof.

2. The method for the treatment of primary biliary cirrhosis according to claim 1 , further comprising administering ursodeoxycholic acid.

3. The method for the treatment of primary biliary cirrhosis according to claim 1 , wherein the (R)-2-[3-[[N-(benzoxazole-2-yl)-N-3-(4-methoxyphenoxy)propyl]aminomethyl]phenoxy] butyric acid, a salt thereof, or a solvate thereof is administered to the patient in a daily dose of 0.05 to 0.8 mg.

4. The method for the treatment of primary biliary cirrhosis according to claim 1 , wherein the administering decreases the level of total bilirubin in the patient.

5. The method for the treatment of primary biliary cirrhosis according to claim 4 , wherein the decrease in the level of total bilirubin in the patient is a decrease of 10% to 75% compared to the level before administration.

Assignments (1)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Feb 26, 2019
From: NAKAMURA, MITSUMASA; KOJIMA, SATOSHI; TANIGAWA, RYOHEI
To: KOWA COMPANY, LTD.
Reel/Frame 048440/0026 →
Continuity (2)
Provisional Application 62463258 · Feb 24, 2017
Related Publication 20180250274A1 · Sep 6, 2018