IP Library Granted Patent US 10,925,886
Granted Patent B2
US 10,925,886 · App. 15/913,541 · Granted Feb 23, 2021

Prevention and treatment of inflammatory conditions

Inventor: Vipin Kumar Chaturvedi (Rancho Sante Fe, CA)
Assignee: GRI BIO, INC.
A61K31/7032A61K31/07A61K31/192A61K31/203A61K31/4436A61K45/06Y02A50/30
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Quick Facts
Patent No.
US 10,925,886
App. No.
15/913,541
Granted
Feb 23, 2021
Kind
B2
Abstract

The present embodiments relate to methods for the prevention and treatment of inflammatory conditions such as alcoholic liver disease (ALD). More specifically the present embodiments relate to the prevention and treatment of ALD through the administration of an Retinoic Acid Receptor (RAR) agonist. Some embodiments relate to use of tazarotene in the prevention and treatment of alcohol-induced liver injury, alcohol-related liver disease, fatty liver disease, hepatic steatosis, alcoholic hepatitis or alcoholic cirrhosis.

Claims (8)

1. A method of treating an inflammatory condition of the liver in a subject in need thereof, the method comprising administering an amount of RARγ-selective agonist sufficient to inhibit activation of pro-inflammatory type I NKT cells to the subject,

wherein the administered RARγ-selective agonist inhibits activation of pro-inflammatory type I NKT cells in the subject, thereby treating the inflammatory condition of the liver.

2. The method of claim 1 , wherein the inflammatory condition of the liver is selected from the group consisting of: fatty liver disease, alcohol induced hepatitis, non-alcoholic steatosis hepatitis, cirrhosis, fulminating cirrhosis, idiopathic hepatitis, viral-induced hepatitis (A, B, C and other), inflammatory hepatitis associated with hepato-biliary carcinoma, ischemic reperfusion injury, and solid organ transplantation.

3. The method of claim 1 , wherein the inflammatory condition of the liver is an alcohol-induced liver injury selected from the group consisting of: alcohol-related liver disease, fatty liver disease, hepatic steatosis, alcoholic hepatitis and alcoholic cirrhosis.

4. The method of claim 1 , wherein the inflammatory condition of the liver is alcoholic liver disease.

5. The method of claim 1 , wherein the inflammatory condition of the liver is hepatic reperfusion injury.

6. The method of claim 1 , wherein the inflammatory condition of the liver is hepatic steatosis.

7. The method of claim 1 , wherein the amount of the RARγ-selective agonist is about 1 mg/day to about 50 mg/day.

Assignments (4)
SECURITY INTEREST Recorded Dec 15, 2022
From: GRI BIO, INC.
To: ALTIUM GROWTH FUND, LP
Reel/Frame 062108/0599 →
SECURITY INTEREST Recorded Nov 2, 2018
From: GRI BIO, INC.
To: TEP BIOTECH, LLC
Reel/Frame 047399/0239 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Mar 9, 2018
From: CHATURVEDI, VIPIN KUMAR
To: GLYCOREGIMMUNE, INC.
Reel/Frame 045159/0631 →
CHANGE OF NAME Recorded Mar 9, 2018
From: GLYCOREGIMMUNE, INC.
To: GRI BIO, INC.
Reel/Frame 045560/0049 →
Continuity (3)
Continuation 14128566
Provisional Application 61501139 · Jun 24, 2011
Related Publication 20180193368A1 · Jul 12, 2018