IP Library Granted Patent US 10,434,107
Granted Patent B2
US 10,434,107 · App. 15/940,941 · Granted Oct 8, 2019

Synthetic bile acid compositions and methods

Inventors: Robert M. Moriarty (Parsippany, NJ); Nathaniel E. David (Parsippany, NJ); Nadir Ahmeduddin Mahmood (Parsippany, NJ)
Assignee: ALLERGAN SALES, LLC
A61K31/575A61K38/08A61K45/06A61K47/24C07J9/00
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Quick Facts
Patent No.
US 10,434,107
App. No.
15/940,941
Granted
Oct 8, 2019
Kind
B2
Abstract

Bile acids and related compositions and methods of synthesis and use. More specifically, deoxycholic acid and related compositions, said compositions being free of all moieties of animal origin and free of pyrogenic moieties.

Claims (10)

1. A method for reducing the appearance of a skin condition in a skin region of a subject in need thereof, the method comprising administering locally to said skin region a composition comprising: a skin-tightening effective amount of DCA

or a pharmaceutically acceptable salt thereof, wherein the DCA comprises a synthetic side chain of formula:

and at least one pharmaceutically acceptable excipient and/or carrier; and wherein the skin condition being reduced is loose skin or wrinkles.

2. The method of claim 1 , wherein the DCA or the pharmaceutically acceptable salt thereof is present in the composition in an amount of about 0.1% w/v to about 2% w/v.

3. The method of claim 1 , wherein the composition further comprises phosphatidylcholine.

4. The method of claim 3 , wherein the phosphatidylcholine is present in the composition in an amount of up to 5% w/v.

5. The method of claim 1 , wherein the composition does not contain phosphatidylcholine.

6. The method of claim 1 , wherein the region of skin is selected from the group consisting of under eye, under chin, under arm, buttock, cheek, brow, calf, back, thigh, ankle, and stomach.

7. The method of claim 1 , wherein the DCA, or a pharmaceutically acceptable salt thereof, is sodium deoxycholate.

8. The method of claim 1 , wherein the administering involves delivering the composition via a subcutaneous or transdermal injection.

Assignments (3)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jul 19, 2021
From: MORIARTY, ROBERT M.; DAVID, NATHANIEL E.; MAHMOOD, NADIR AHMEDUDDIN
To: KYTHERA BIOPHARMACEUTICALS, INC.
Reel/Frame 056904/0887 →
MERGER AND CHANGE OF NAME Recorded Aug 7, 2019
From: KYTHERA BIOPHARMACEUTICALS, LLC; ALLERGAN SALES, LLC
To: ALLERGAN SALES, LLC
Reel/Frame 049981/0649 →
CHANGE OF NAME Recorded Aug 3, 2019
From: KYTHERA BIOPHARMACEUTICALS, INC.
To: KYTHERA BIOPHARMACEUTICALS, LLC
Reel/Frame 049951/0872 →
Continuity (7)
Continuation 15349573 · Nov 11, 2016
Continuation 14503273 · Sep 30, 2014
Continuation 13741212 · Jan 14, 2013
Continuation 12035339 · Feb 21, 2008
Provisional Application 60956875 · Aug 20, 2007
Provisional Application 60945035 · Jun 19, 2007
Related Publication 20180221391A1 · Aug 9, 2018