IP Library Granted Patent US 10,953,007
Granted Patent B2
US 10,953,007 · App. 15/994,235 · Granted Mar 23, 2021

Compounds useful as modulators of TRPM8

Inventors: Chad Priest (Leucadia, CA); Alain Noncovich (San Diego, CA); Andrew Patron (San Marcos, CA); Jane Ung (San Diego, CA)
Assignee: Firmenich Incorporated
A61K31/497A01N37/18A01N43/10A01N43/40A01N43/56A01N43/60A01N43/76A01N43/78A01N43/80A01N43/90A23L27/88A23L33/10A61K8/42A61K8/49A61K8/494A61K8/4926A61K8/4973A61K8/4986A61K8/69A61K31/165A61K31/381A61K31/415A61K31/4155A61K31/422A61K31/426A61K31/437A61K31/4409A61K31/4436A61Q19/00C07C233/11C07C235/20C07C235/24C07C235/34C07D213/40C07D213/75C07D231/40C07D277/28C07D307/52C07D333/20C07D333/24C07D333/32C07D405/12C07D407/12C07D409/12C07D409/14C07D413/12C07D417/12C07D471/04A23V2002/00A61K2800/10A61K2800/40A61Q1/02A61Q5/02A61Q5/12A61Q9/02A61Q11/00A61Q15/00A61Q17/02A61Q17/04A61Q19/001A61Q19/10C07C2601/14
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Quick Facts
Patent No.
US 10,953,007
App. No.
15/994,235
Granted
Mar 23, 2021
Kind
B2
Abstract

The present invention includes compounds useful as modulators of TRPM8, such as compounds of Formula (I) and the subgenus and species thereof; personal products containing those compounds; and the use of those compounds and the personal products, particularly the use of increasing or inducing chemesthetic sensations, such as cooling or cold sensations.

Claims (16)

1. A composition comprising a compound having a structure of

or a salt or solvate thereof.

2. The composition of claim 1 , wherein the composition is an ingestible composition or personal care composition.

3. The composition of claim 1 , wherein the composition is in the form of a solid, semi-solid, plaster, solution, suspension, lotion, cream, foam, gel, paste, emulsion, or a combination thereof.

4. The composition of claim 1 , wherein the compound in the composition is in a concentration ranging from about 0.0001 ppm to 100,000 ppm.

5. A composition comprising a compound having a structure of

or a salt or solvate thereof.

6. The composition of claim 5 , wherein the composition is an ingestible composition or personal care composition.

7. The composition of claim 5 , wherein the composition is in the form of a solid, semi-solid, plaster, solution, suspension, lotion, cream, foam, gel, paste, emulsion, or a combination thereof.

8. The composition of claim 5 , wherein the compound in the composition is in a concentration ranging from about 0.0001 ppm to 100,000 ppm.

9. A composition comprising a compound having a structure of

or a salt or solvate thereof.

10. The composition of claim 9 , wherein the composition is an ingestible composition or personal care composition.

11. The composition of claim 9 , wherein the composition is in the form of a solid, semi-solid, plaster, solution, suspension, lotion, cream, foam, gel, paste, emulsion, or a combination thereof.

12. The composition of claim 9 , wherein the compound in the composition is in a concentration ranging from about 0.0001 ppm to 100,000 ppm.

13. A composition comprising a compound, wherein the wherein the concentration of the compound in the composition ranges from 0.0001 ppm to 100,000 ppm; and wherein the compound is a compound of one of the following chemical formulae:

Assignments (2)
MERGER Recorded Oct 16, 2019
From: SENOMYX, INC.
To: FIRMENICH INCORPORATED
Reel/Frame 050733/0195 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Apr 10, 2019
From: PRIEST, CHAD; NONCOVICH, ALAIN; PATRON, ANDREW; UNG, JANE
To: SENOMYX, INC.
Reel/Frame 048846/0931 →
Continuity (5)
Continuation 15205608 · Jul 8, 2016
Continuation 13883349
Provisional Application 61443490 · Feb 16, 2011
Provisional Application 61410634 · Nov 5, 2010
Related Publication 20180289704A1 · Oct 11, 2018