IP Library Granted Patent US 11,376,235
Granted Patent B2
US 11,376,235 · App. 16/076,092 · Granted Jul 5, 2022

Inhibitor of inflammasome activation

Inventors: Shimpei Watanabe (Tokyo, JP); Ayako Arai (Tokyo, JP); Yuichi Takajo (Tokyo, JP); Satoshi Inamasu (Tokyo, JP); Satoshi Yomoda (Tokyo, JP); Akiko Ohno (Tokyo, JP); Yuko Kitahara (Tokyo, JP); Taisaku Kanatani (Tokyo, JP)
Assignee: KRACIE HOLDINGS, LTD.
A61K31/365A23L33/105A61K8/49A61K8/4973A61K8/602A61K8/97A61K8/9789A61K31/7048A61K36/28A61K36/634A61P1/16A61P3/04A61P3/10A61P9/00A61P9/10A61P13/12A61P17/00A61P17/06A61P17/10A61P17/14A61P25/16A61P25/28A61P27/02A61P29/00A61Q19/00A23V2002/00A23V2200/30A23V2250/21
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Quick Facts
Patent No.
US 11,376,235
App. No.
16/076,092
Granted
Jul 5, 2022
Kind
B2
Abstract

To provide a novel inflammasome inhibitor capable of inhibiting activation of inflammasome, the present inventors newly found that arctigenin reduces the amount of 1L-1β released and the amount of activated caspase-1 upon stimulation with ATP, palmitic acid, MSU and Poly(dA:dT) and thus has an effect of inhibiting inflammasome activation. The present invention provides an inhibitor of inflammasome activation that comprises arctigenin as an active ingredient.

Claims (2)

1. A method for treating or improving non-alcoholic steatohepatitis (NASH) through inhibition of inflammasome activation including administering arctigenin and/or arctiin to a subject in need thereof, wherein arctigenin and/or arctiin inhibits release of inflammatory cytokines as IL-1αa, IL-1β, IL-6, IL-18, IL-33, TNF-α, and HMGB1 in the subject after administration.

2. The method for inhibiting inflammasome activation according to claim 1 , wherein only arctiin is administered to the subject.

Assignments (2)
CHANGE OF NAME Recorded Jun 13, 2024
From: KRACIE HOLDINGS, LTD.
To: KRACIE, LTD.
Reel/Frame 067714/0179 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Aug 7, 2018
From: WATANABE, SHIMPEI; ARAI, AYAKO; TAKAJO, YUICHI; INAMASU, SATOSHI; YOMODA, SATOSHI; OHNO, AKIKO; KITAHARA, YUKO; KANATANI, TAISAKU
To: KRACIE HOLDINGS, LTD.
Reel/Frame 046574/0015 →
Priority Claims (1)
JP JP2016-021844 · Feb 8, 2016 · national
Continuity (1)
Related Publication 20190099400A1 · Apr 4, 2019