IP Library › Granted Patent US 10,906,909
Granted Patent B2
US 10,906,909 · App. 16/086,053 · Granted Feb 2, 2021

Treatment of cognitive and mood symptoms in neurodegenerative and neuropsychiatric disorders with ALPHA5-containing GABAA receptor agonists

Inventors: James M. Cook (Milwaukee, WI); Guanguan Li (Milwaukee, WI); Michael Ming-Jin Poe (Vernon, CT); Miroslav M. Savic (Belgrade, RS); Etienne Sibille (Toronto, CA)
Assignees: UWM Research Foundation, Inc.; Centre for Addiction and Mental Health; University of Belgrade—Faculty of Pharmacy
C07D487/04A61P25/22
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Quick Facts
Patent No.
US 10,906,909
App. No.
16/086,053
Granted
Feb 2, 2021
Kind
B2
Abstract

Provided herein are alpha5-containing GABA A receptor agonists and pharmaceutical compositions and methods of treatment of cognitive and mood symptoms in neurodegenerative and neuropsychiatric disorders using them.

Claims (11)

1. A compound selected from the group consisting of:

or a pharmaceutically acceptable salt thereof.

2. The compound of claim 1 that is

or a pharmaceutically acceptable salt thereof.

3. The compound of claim 1 that is

or a pharmaceutically acceptable salt thereof.

4. The compound of claim 1 that is

or a pharmaceutically acceptable salt thereof.

5. A pharmaceutical composition comprising the compound according to claim 2 , or a pharmaceutically acceptable salt thereof, and a pharmaceutically acceptable excipient.

6. A pharmaceutical composition comprising the compound according to claim 3 , or a pharmaceutically acceptable salt thereof, and a pharmaceutically acceptable excipient.

7. A pharmaceutical composition comprising the compound according to claim 4 , or a pharmaceutically acceptable salt thereof, and a pharmaceutically acceptable excipient.

Assignments (3)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Nov 11, 2020
From: COOK, JAMES M.; LI, GUANGUAN; POE, MICHAEL MING-JIN
To: UWM RESEARCH FOUNDATION, INC.
Reel/Frame 054339/0506 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Nov 5, 2020
From: SAVIC, MIROSLAV M.
To: UNIVERSITY OF BELGRADE - FACULTY OF PHARMACY
Reel/Frame 054283/0410 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Nov 5, 2020
From: SIBILLE, ETIENNE
To: CENTRE FOR ADDICTION AND MENTAL HEALTH
Reel/Frame 054283/0562 →
Continuity (2)
Provisional Application 62310409 · Mar 18, 2016
Related Publication 20200181146A1 · Jun 11, 2020
Cited By (1)
US 12,636,291