IP Library Granted Patent US 10,765,744
Granted Patent B2
US 10,765,744 · App. 16/093,370 · Granted Sep 8, 2020

Magnetic particle conjugates, micelles, and methods of delivering agents

Inventors: Carlos Rinaldi (Gainesville, FL); Sun Hao (Wilmette, IL); Brent S. Sumerlin (Gainesville, FL)
Assignee: University of Florida Research Foundation, Inc.
A61K41/0028A61K9/1075A61K47/02A61K47/34A61K47/52A61K47/60A61K47/6907A61K47/6923
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Quick Facts
Patent No.
US 10,765,744
App. No.
16/093,370
Granted
Sep 8, 2020
Kind
B2
Abstract

Embodiments of the present disclosure provide for magnetic particle conjugates, methods of making the magnetic particle conjugates, methods of using magnetic particle conjugates, micelles (also referred to as a “magnetic composite nanocarrier” (MC-NC)), methods of making micelles, methods of using micelles, and the like.

Claims (13)

1. A composition comprising: a magnetic particle conjugate having a magnetic particle and a polymer attached to the magnetic particle, wherein the polymer includes an agent (A gent ) bonded to the polymer through thermally degradable retro-Diels-Alder-agent group, wherein the polymer comprises:

wherein w is 1 to 20, x is 0 to 20, y is 0 to 60, and z is 0 to 10, wherein the polymer is bonded to the magnetic particle on the left of the structure.

2. The composition of claim 1 , wherein the magnetic particle is a material represented by M a x M b (1-x) Fe 2 O 4 , where each of M a and M b are independently selected from Fe, Co, Mn, Zn, Ta, Sr, or Ni, wherein x is 0 to 1, wherein M a and M b are different metals.

3. The composition of claim 2 , wherein the magnetic particle is a material selected from the group consisting of: Fe 3 O 4 , γFe 2 O 3 , αFe 2 O 3 , MnFe 2 O 4 , ZnFe 2 O 4 , or Mn 0.5 Zn 0.5 Fe 2 O 4 .

4. The composition of claim 1 , wherein w is 14, x is 11, y is 40 and z is 10.

5. The composition of claim 1 , wherein the agent includes a drug, a therapeutic agent, a radiological agent, or a biological agent.

6. The composition of claim 1 , wherein the polymer fully encapsulates both the agent and the magnetic particles.

7. A composition, comprising:

a micelle including a plurality a magnetic particle conjugate having a magnetic particle and a polymer attached to the magnetic particle, wherein the polymer has a hydrophobic region and a hydrophilic region, wherein the hydrophobic region of the polymer is located in a central region of the micelle and the hydrophilic region is located away from the central region and forms the micelle outer boundary, wherein the polymer includes an agent (A gent ) bonded to the polymer through thermally degradable retro-Diels-Alder-agent group, wherein the polymer comprises:

wherein w is 1 to 20, x is 0 to 20, y is 0 to 60, and z is 0 to 10, wherein the polymer is bonded to the magnetic particle on the left of the structure.

8. The composition of claim 7 , wherein the magnetic particle is a material selected from the group consisting of: Fe 3 O 4 , γFe 2 O 3 , αFe 2 O 3 , and MnFe 2 O 4 , ZnFe 2 O 4 , or Mn 0.5 Zn 0.5 Fe 2 O 4 .

9. The composition of claim 7 , wherein the micelle in encapsulated using a hydrophobic block copolymer that has thermally labile backbone bonds.

10. The composition of claim 7 , further comprising a targeting agent.

Assignments (2)
CONFIRMATORY LICENSE Recorded Mar 26, 2020
From: UNIVERSITY OF FLORIDA
To: NATIONAL SCIENCE FOUNDATION
Reel/Frame 052249/0791 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Feb 14, 2019
From: RINALDI, CARLOS; HAO, SUN; SUMERLIN, BRENT S.
To: UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INC.
Reel/Frame 048335/0644 →
Continuity (2)
Provisional Application 62328053 · Apr 27, 2016
Related Publication 20190290761A1 · Sep 26, 2019