IP Library Granted Patent US 10,287,353
Granted Patent B2
US 10,287,353 · App. 16/103,865 · Granted May 14, 2019

Combination therapies of HDAC inhibitors and PD-1 inhibitors

Inventors: Reid P. Bissonnette (Carlsbad, CA); Alain Rolland (San Diego, CA); Mireille Gillings (Las Vegas, NV)
Assignee: HUYA Bioscience International, LLC
C07K16/2818A61K31/167A61K31/18A61K31/343A61K31/395A61K31/4045A61K31/4184A61K31/4406A61K31/506A61K38/15A61K39/39541A61K39/39558A61K45/06A61K2039/505A61K2039/545C07K2317/76
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Quick Facts
Patent No.
US 10,287,353
App. No.
16/103,865
Granted
May 14, 2019
Kind
B2
Abstract

Provided herein are combinations that include an HDACi and a PD-1 inhibitor that are useful for treating cancer, including reducing and/or preventing cancer metastasis. The combination is also useful for treating cancer that has been previously treated with a PD-L1 inhibitor.

Claims (7)

1. A method for treating melanoma in a subject, comprising administering to said subject a therapeutically effective amount of a compound of the following formula:

in combination with nivolumab, wherein the subject has been treated with a PD-L1 checkpoint inhibitor.

2. The method of claim 1 , wherein the compound is administered at an amount of about 30 mg BIW.

3. The method of claim 1 , wherein nivolumab is administered as an intravenous infusion over about 30 minutes.

4. The method of claim 1 , wherein the melanoma is Stage II, III or IV melanoma.

5. The method of claim 1 , wherein the melanoma is resistant/refractory melanoma.

6. The method of claim 1 , wherein the melanoma is metastatic.

Assignments (3)
SECURITY INTEREST Recorded Feb 21, 2024
From: HUYABIO INTERNATIONAL, LLC
To: R-BRIDGE INVESTMENT SIX PTE. LTD.
Reel/Frame 066515/0036 →
CHANGE OF NAME Recorded Nov 9, 2021
From: HUYA BIOSCIENCE INTERNATIONAL, LLC
To: HUYABIO INTERNATIONAL, LLC
Reel/Frame 058079/0643 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Oct 7, 2020
From: BISSONNETTE, REID P.; ROLLAND, ALAIN; GILLINGS, MIREILLE
To: HUYA BIOSCIENCES INTERNATIONAL, LLC
Reel/Frame 054001/0023 →
Continuity (4)
Continuation 15592988 · May 11, 2017
Provisional Application 62436361 · Dec 19, 2016
Provisional Application 62335044 · May 11, 2016
Related Publication 20180355042A1 · Dec 13, 2018
Cited By (2)
US 12,258,323 US 12,427,153