IP Library Granted Patent US 10,758,553
Granted Patent B2
US 10,758,553 · App. 16/125,511 · Granted Sep 1, 2020

Antibacterial use of halogenated salicylanilides

Inventors: Emilie Flora Aurore Delavenne (Le Mans, FR); Daniel Jean Jacques Simon (Søborg, DK); Morten Otto Alexander Sommer (Virum, DK); Rasmus Vendler Toft-Kehler (Copenhagen Ø, DK)
Assignee: UNION therapeutics A/S
A61K31/609A61K9/0014A61K9/06A61K47/10A61K47/14A61K47/26A61P17/00A61P31/04
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Quick Facts
Patent No.
US 10,758,553
App. No.
16/125,511
Granted
Sep 1, 2020
Kind
B2
Abstract

The invention relates to a halogenated salicylanilide selected from closantel, rafoxanide, oxyclozanide and niclosamide and derivatives thereof including salts, hydrates, esters and the like for use in the topical treatment or prevention of infections caused by Gram-positive bacteria such as Staphylococcus , in particular Staphylococcus aureus , and Streptococcus , in particular Streptococcus pyogenes . Grain positive bacteria treated with the halogenated salicylanilides exhibit a very low frequency of appearance of resistant mutants compared to commonly used topical antibiotics.

Claims (21)

1. A method of treating pyoderma in a non-human animal, the method comprising topically administering to said non-human animal an effective amount of oxyclozanide.

2. The method of claim 1 , wherein the animal is a companion animal.

3. The method of claim 1 , wherein the animal is a dog or cat.

4. The method of claim the method of claim 1 , wherein the pyoderma is caused by Staphylococcus spp.

5. The method of claim the method of claim 1 , wherein the pyoderma is caused by Staphylococcus aureus.

6. The method of claim 1 , wherein the non-human animal is a dog.

7. The method of claim 1 , wherein the oxyclozanide is topically administered to said non-human animal in the form of a pharmaceutical composition comprising from 1% to 20% by weight oxyclozanide.

8. The method of claim 1 , wherein the oxyclozanide is topically administered to said non-human animal in the form of a pharmaceutical composition comprising from 2% to 20% by weight oxyclozanide.

9. The method of claim 1 , wherein the oxyclozanide is topically administered to said non-human animal in the form of a pharmaceutical composition comprising from 2% to 10% by weight oxyclozanide.

10. The method of claim 1 , wherein the oxyclozanide is topically administered to said non-human animal in the form of an epicutaneous pharmaceutical composition.

11. The method of claim 1 , wherein the oxyclozanide is topically administered to said non-human animal in the form of a pharmaceutical composition selected from a cream, a foam, a gel, droplets, a lotion and an ointment.

12. The method of claim 1 , wherein the oxyclozanide is topically administered to said non-human animal once per day.

13. A method of treating pyoderma in a dog, the method comprising topically administering to said dog an effective amount of oxyclozanide.

14. The method of claim 13 , wherein the pyoderma is caused by Staphylococcus spp.

15. The method of claim 13 , wherein the pyoderma is caused by Staphylococcus aureus.

16. The method of claim 13 , wherein the oxyclozanide is topically administered to said dog in the form of a pharmaceutical composition comprising from 1% to 20% by weight oxyclozanide.

17. The method of claim 13 , wherein the oxyclozanide is topically administered to said dog in the form of a pharmaceutical composition comprising from 2% to 20% by weight oxyclozanide.

18. The method of claim 13 , wherein the oxyclozanide is topically administered to said dog in the form of a pharmaceutical composition comprising from 2% to 10% by weight oxyclozanide.

19. The method of claim 13 , wherein the oxyclozanide is topically administered to said dog in the form of an epicutaneous pharmaceutical composition.

20. The method of claim 13 , wherein the oxyclozanide is topically administered to said dog in the form of a pharmaceutical composition selected from a cream, a foam, a gel, droplets, a lotion and an ointment.

21. The method of claim 13 , wherein the oxyclozanide is topically administered to said dog once per day.

Assignments (4)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jul 22, 2020
From: DELAVENNE, EMILIE FLORA AURORE; SIMON, DANIEL JEAN JACQUES; SOMMER, MORTEN OTTO ALEXANDER; TOFT-KEHLER, RASMUS VENDLER
To: ANTIBIOTX APS
Reel/Frame 053279/0085 →
CHANGE OF NAME Recorded Jul 22, 2020
From: ANTIBIOTX APS
To: ANTIBIOTX A/S
Reel/Frame 053279/0319 →
CORRECTIVE ASSIGNMENT TO CORRECT THE ASSIGNEE PREVIOUSLY RECORDED ON REEL 049069 FRAME 0481. ASSIGNOR(S) HEREBY CONFIRMS THE CHANGE OF NAME. Recorded Jan 16, 2020
From: ANTIBIOTX A/S
To: UNION THERAPEUTICS A/S
Reel/Frame 051620/0491 →
CHANGE OF NAME Recorded Dec 18, 2018
From: ANTIBIOTX A/S
To: UNION THERAPEUTICS
Reel/Frame 049069/0481 →
Priority Claims (1)
SE 1451054 · Sep 12, 2014 · national
Continuity (2)
Continuation 15510304
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