IP Library Granted Patent US 10,652,527
Granted Patent B2
US 10,652,527 · App. 16/189,551 · Granted May 12, 2020

Goggle imaging systems and methods

Inventor: Samuel Achilefu (St. Louis, MO)
Assignee: Washington University
H04N13/344A61B34/25A61B90/30A61B90/36A61B90/361A61K49/0032A61K49/0034A61K49/0056C07K7/06G02B27/017H04N5/374A61B1/0005A61B1/0692A61B2090/364
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Quick Facts
Patent No.
US 10,652,527
App. No.
16/189,551
Granted
May 12, 2020
Kind
B2
Abstract

A compound of formula (I) is provided having the structure: cypate-cyclo(Cys-Gly-Arg-Asp-Ser-Pro-Cys)-Lys-OH, and each amino acid is independently in a D or L configuration. Also provided are pharmaceutical compositions that include the compound of formula (I) and its use in treating cancer by administering it to a patient in need thereof.

Claims (13)

1. A compound of formula (I), or a salt thereof,

cypate-cyclo(Cys-Gly-Arg-Asp-Ser-Pro-Cys)-Lys-OH  (I)

wherein each amino acid is independently in a D or L configuration.

2. The compound according to claim 1 , wherein the cypate is

3. The compound of formula (I) according to claim 1 , wherein at least one of the Cys amino acid residues is D-Cys.

4. The compound of formula (I) according to claim 1 having the formula:

5. The compound of formula (I) according to claim 1 , wherein the compound is LS-301:

6. A pharmaceutical composition comprising:

the compound of formula (I) according to claim 1 , or a pharmaceutically acceptable salt thereof, and

a pharmaceutically acceptable carrier.

7. The pharmaceutical composition according to claim 6 , wherein said composition is in a formulation suitable for intravenous administration.

8. The pharmaceutical composition according to claim 6 , wherein the compound is LS-301.

9. The compound of formula (I) according to claim 1 , wherein the compound is

Assignments (2)
CONFIRMATORY LICENSE Recorded May 28, 2020
From: WASHINGTON UNIVERSITY
To: NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT
Reel/Frame 052774/0697 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Nov 19, 2018
From: ACHILEFU, SAMUEL; CULVER, JOSEPH; AKERS, WALTER; BAUER, ADAM; GRUEV, VIKTOR; LIU, YANG
To: WASHINGTON UNIVERSITY
Reel/Frame 047544/0703 →
Continuity (3)
Continuation 14374002
Provisional Application 61589623 · Jan 23, 2012
Related Publication 20190104300A1 · Apr 4, 2019
Cited By (1)
US 12,238,268