IP Library Granted Patent US 10,980,741
Granted Patent B2
US 10,980,741 · App. 16/210,896 · Granted Apr 20, 2021

Compositions and methods for treating pterygium recurrence

Inventor: Jinsong Ni (Irvine, CA)
Assignee: Cloudbreak Therapeutics, LLC
A61K9/0048A61F9/00A61F9/0017A61K9/0051A61K9/06A61K9/08A61K9/10A61K9/107A61K31/404A61K31/407A61K31/496A61K45/06A61K47/26A61P27/00A61P27/02
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Quick Facts
Patent No.
US 10,980,741
App. No.
16/210,896
Granted
Apr 20, 2021
Kind
B2
Abstract

Compositions and methods for inducing pterygium regression from visual axis/central cornea, stabilizing pterygium, treating hyperemia and symptoms in pterygium patients, and treating pterygium recurrence following pterygiectomy are disclosed. The methods include administration of a multikinase inhibitor, an antimetabolite or a combination thereof to patients in need thereof.

Claims (19)

1. A method for treating pterygium in an eye of a subject, comprising administering to the affected eye of the subject a therapeutically effective amount of nintedanib.

2. The method of claim 1 , wherein treating pterygium comprises reducing hyperemia, regressing a pterygium, or stabilizing a pterygium.

3. The method of claim 2 , wherein treating pterygium comprises reducing hyperemia.

4. The method of claim 2 , wherein treating pterygium comprises pterygium regression.

5. The method of claim 2 , wherein treating pterygium comprises pterygium stabilization.

6. The method of claim 2 , wherein treating pterygium further comprises reducing a symptom of pterygium.

7. The method of claim 6 , wherein the symptom of pterygium comprises ocular discomfort, irritation, blurred vision, foreign body sensation, or pain.

8. The method of claim 6 , wherein the symptom of pterygium is a clinical symptom or a subclinical symptom.

9. The method of claim 1 , wherein the nintedanib is administered to the affected eye in the form of a topical ocular formulation or an ocular implant.

10. The method of claim 9 , wherein the topical ocular formulation is a solution or a suspension.

11. The method of claim 9 , wherein the topical ocular formulation further comprises one or more pharmaceutically acceptable excipients.

12. The method of claim 9 , wherein the ocular implant is injected into the affected eye.

13. The method of claim 9 , wherein the ocular implant further comprises one or more pharmaceutically acceptable excipients.

14. The method of claim 1 , further comprising administering to the affected eye of the subject a pharmaceutically effective amount of an antimetabolite.

15. The method of claim 14 , wherein the antimetabolite blocks epithelial and fibroblast cell proliferation.

16. The method of claim 14 , wherein the antimetabolite is selected from the group consisting of mitomycin C, 5-fluorouracil, and thiotepa.

17. The method of claim 1 , wherein the administration is performed prior to surgical removal of a pterygium.

18. The method of claim 1 , wherein the administration is performed during a surgical procedure to remove a pterygium.

19. The method of claim 1 , wherein the administration is performed following surgical removal of a pterygium.

Assignments (1)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Oct 3, 2019
From: NI, JINSONG
To: CLOUDBREAK THERAPEUTICS, LLC
Reel/Frame 050618/0716 →
Continuity (7)
Continuation 15991698 · May 29, 2018
Continuation 15474620 · Mar 30, 2017
Continuation 15375820 · Dec 12, 2016
Continuation PCTUS2016035726 · Jun 3, 2016
Provisional Application 62172063 · Jun 6, 2015
Provisional Application 62186660 · Jun 30, 2015
Related Publication 20190110984A1 · Apr 18, 2019
Cited By (3)
US 12,186,424 US 12,491,183 US 12,589,025