IP Library Granted Patent US 10,472,632
Granted Patent B2
US 10,472,632 · App. 16/241,943 · Granted Nov 12, 2019

Anti-connexin compounds targeted to connexins and methods of use thereof

Inventors: Wilda Laux (Mangere, NZ); Colin Richard Green (Auckland, NZ)
Assignee: OCUNEXUS THERAPEUTICS, INC.
C12N15/113A61K31/711A61K31/7105C12N15/111C12N15/1138C12N2310/11C12N2310/12C12N2310/315C12N2320/31Y02P20/582
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Quick Facts
Patent No.
US 10,472,632
App. No.
16/241,943
Granted
Nov 12, 2019
Kind
B2
Abstract

Methods and compositions for modulating the activities of connexins are provided, including, for example, for use in post-surgical, trauma, or tissue engineering applications. These compounds and methods can be used therapeutically, for example, to reduce the severity of adverse effects associated diseases and disorders where localized disruption in direct cell-cell communication is desirable.

Claims (12)

1. A method for treating a subject for corneal trauma, comprising topically administering to the eye of said subject a composition comprising a pluronic F127 gel, phosphate buffered saline, and a connexin 43-downregulating amount of a connexin 43 antisense compound, wherein said connexin 43 antisense compound is 5′ GTA ATT GCG GCA AGA ATT GTT TCT GTC 3′ (SEQ ID NO: 1).

2. The method of claim 1 , wherein said trauma is a penetrating eye trauma.

3. A method of claim 2 wherein the eye trauma is chemical trauma.

4. A method of claim 2 wherein the eye trauma is mechanical trauma.

5. A method of claim 1 wherein the eye trauma results in corneal epithelial damage.

6. A method of claim 1 wherein the connexin 43 antisense compound is administered to a subject having an amniotic membrane graft.

7. A method of claim 1 wherein said composition comprises 30% (w/w) pluronic F127 gel in phosphate buffered saline.

8. A method of claim 1 wherein the pluronic gel comprises up to 15% (w/w) pluronic F127, up to 20% (w/w) pluronic F127, up to 25% (w/w) pluronic F127 or up to 30% (w/w) pluronic F127 in phosphate buffered saline.

9. A method of claim 1 wherein the composition further comprises a preservative.

10. A method of claim 1 wherein the composition is administered once.

11. A method of claim 1 wherein the composition is administered more than once.

12. A method of claim 1 wherein the subject is a human.

Assignments (3)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Feb 1, 2019
From: LAUX, WILDA; GREEN, COLIN
To: CODA THERAPEUTICS (NZ) LTD
Reel/Frame 048223/0302 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Feb 1, 2019
From: CODA THERAPEUTICS (NZ) LTD
To: CODA THERAPEUTICS, INC.
Reel/Frame 048226/0321 →
CHANGE OF NAME Recorded Feb 1, 2019
From: CODA THERAPEUTICS, INC.
To: OCUNEXUS THERAPEUTICS, INC.
Reel/Frame 048230/0135 →
Priority Claims (1)
NZ 529936 · Dec 3, 2003 · national
Continuity (4)
Division 14467978 · Aug 25, 2014
Division 13230744 · Sep 12, 2011
Division 10581813
Related Publication 20190194657A1 · Jun 27, 2019
Cited By (1)
US 12,667,586