IP Library Granted Patent US 12,396,980
Granted Patent B2
US 12,396,980 · App. 16/298,824 · Granted Aug 26, 2025

Melatonin for preventing and treating radiation cystitis

Inventors: Lasse Lindblad (Ålsgårde, DK); Lars Otto Uttenthal (Madrid, ES)
Assignee: REPOCEUTICALS A/S
A61K31/4045A61K9/08A61K31/122A61K31/167A61K31/355A61K31/375A61K31/385A61K47/20
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Quick Facts
Patent No.
US 12,396,980
App. No.
16/298,824
Granted
Aug 26, 2025
Kind
B2
Abstract

Compositions comprising melatonin and/or derivatives thereof are provided for topical administration to the epithelium of the urinary bladder by instillation into the bladder to protect against or treat bladder injury due to irradiation and/or cytotoxic agents.

Claims (14)

1. A method for reducing urinary bladder injury selected from radiation cystitis caused by irradiation by pelvic external beam radiotherapy and/or irradiation by pelvic brachyradiotherapy, comprising:

(a) administering a composition consisting of melatonin, dimethyl sulfoxide (DMSO), water and optionally sodium chloride directly into the urinary bladder of a subject; and

(b) administering a treatment to the subject, wherein the treatment comprises: radiation treatment to the subject by pelvic external beam radiotherapy and/or pelvic brachyradiotherapy;

wherein administering step (a) is done within one hour before administering step (b) and at intervals after step (b).

2. The method of claim 1 , wherein the radiation cystitis is exacerbated by additional treatment of the subject with a dose of one or more cytotoxic agents.

3. The method of claim 1 , wherein the melatonin is formulated as a solution in dimethyl sulfoxide (DMSO) and diluted in an aqueous medium prior to use.

4. The method of claim 3 , wherein the concentration of dimethyl sulfoxide (DMSO) in the solution is between 100 parts of dimethyl sulfoxide to 300 parts of water by volume and 100 parts of dimethyl sulfoxide to 30 parts of water by volume.

5. The method of claim 1 , wherein the composition is administered 1, 2, 3, or 4 times per day.

6. The method of claim 1 , wherein the composition is administered over a period of up to 3 months.

7. The method of claim 6 , wherein the composition is administered over a period of up to 12 months.

8. The method of claim 1 , wherein a single standard dose of melatonin is 1 mg to 500 mg.

9. The method of claim 8 , wherein the daily dose of the composition is from one to four times the single standard dose.

10. The method of claim 1 , wherein the composition is administered directly into the urinary bladder within 30 minutes before the treatment of (b) is administered to the subject, and at intervals thereafter.

11. The method of claim 1 , wherein the composition consists of 10 mL to 50 mL of DMSO, 25 mg to 250 mg of melatonin, water, and optionally sodium chloride.

Assignments (2)
CHANGE OF NAME Recorded Jan 26, 2022
From: REPOCEUTICALS APS
To: REPOCEUTICALS A/S
Reel/Frame 058869/0645 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Mar 12, 2019
From: LINDBLAD, LASSE; UTTENTHAL, LARS OTTO
To: REPOCEUTICALS APS
Reel/Frame 048579/0927 →
Priority Claims (1)
DK PA201570145 · Mar 13, 2015 · national
Continuity (2)
Continuation 15557044
Related Publication 20200197367A1 · Jun 25, 2020
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