IP Library Granted Patent US 10,703,711
Granted Patent B2
US 10,703,711 · App. 16/350,344 · Granted Jul 7, 2020

Small molecule drugs and related methods for treatment of diseases related to Aβ42 oligomer formation

Inventors: Ambuj K. Singh (Santa Barbara, CA); Christian A. Lang (Santa Barbara, CA)
Assignee: Acelot, Inc.
C07C233/43A61K31/131A61K31/135A61K31/137C07C211/27C07C211/28C07C211/29C07C217/60C07C223/02C07C271/18C07D207/06C07D295/135C07D295/15C07D319/18C07D413/06
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Quick Facts
Patent No.
US 10,703,711
App. No.
16/350,344
Granted
Jul 7, 2020
Kind
B2
Abstract

The present invention provides small molecule drugs and pharmaceutical compositions for the treatment and prevention of diseases related to the formation of Aβ42 oligomers in a subject. It further provides a method of reducing formation of or disrupting Aβ42 oligomers in a subject, the method comprising the step of administering to the subject in need thereof a therapeutically effective amount of a pharmaceutical composition.

Claims (7)

1. A method of reducing formation of or disrupting Aβ42 oligomers in a subject, the method comprising the step of administering to the subject in need thereof a therapeutically effective amount of a pharmaceutical composition comprising a compound selected from the group consisting of AC0101, AC0102, AC0103, AC0104, AC0105, AC0106, AC0107, Benzald1, Fluorophenyl, Aminofluorophenyl and Dimethoxy.

2. The method of claim 1 , wherein the Aβ42 oligomer is a hexamer, dodecamer or high order oligomer and formation of or the amount of the Aβ42 hexamer, oligomer or highly ordered oligomer is reduced.

3. The method of claim 1 , wherein administration of the pharmaceutical composition results in improved or enhanced cognitive function in a subject with decreased cognitive function.

4. The method of claim 1 , wherein the subject is diagnosed with AD.

5. The method of claim 1 , wherein the subject is genetically predisposed to AD.

6. The method of claim 1 , wherein the subject has the gene for early onset familial AD.

7. The method of claim 1 , wherein the subject is at risk for developing AD.

Assignments (1)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jun 4, 2019
From: SINGH, AMBUJ K.; LANG, CHRISTIAN A.
To: ACELOT, INC.
Reel/Frame 049344/0536 →
Continuity (2)
Provisional Application 62707516 · Nov 6, 2017
Related Publication 20190210959A1 · Jul 11, 2019
Cited By (4)
US 12,312,296 US 12,343,319 US 12,344,570 US 12,351,537