IP Library Granted Patent US 11,813,309
Granted Patent B2
US 11,813,309 · App. 16/366,898 · Granted Nov 14, 2023

Method of alleviating chronic wounds

Inventor: Lars Heslet (Gentofte, DK)
Assignee: Reponex Pharmaceuticals APS
A61K38/193A61K31/7024A61K31/728A61K47/26A61K9/0014A61K9/10A61K47/24A61K47/36
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Quick Facts
Patent No.
US 11,813,309
App. No.
16/366,898
Granted
Nov 14, 2023
Kind
B2
Abstract

The present invention provides compositions comprising granulocyte-macrophage colony-stimulating factor (GM-CSF), sucrose octasulfate or sucralfate and hyaluronic acid for the treatment, pre-emptive treatment or prophylaxis of ulcers, wounds and other injuries to the skin or membranes of the body. Other aspects of the invention are methods of treatment or prevention using the compositions described, as well as an application device for use in the methods provided.

Claims (24)

1. A method of alleviating a chronic wound in a subject comprising administering topically to the wound a composition formulated as a hydrogel, the composition comprising:

a granulocyte-macrophage colony-stimulating factor (GM-CSF) having at least 95% sequence identity to SEQ ID. No. 2 at a concentration of 10 μg/g to 300 μg/g;

sucralfate at a concentration of 5% w/w to 20% w/w; and

a salt of hyaluronan at a concentration of 0.1% w/w to 10% w/w.

2. The method of claim 1 , wherein the GM-CSF has a T1151 substitution, wherein the substitution is positioned in accordance with the amino acid positions set forth in SEQ ID No. 1.

3. The method of claim 1 , wherein the GM-CSF has a 1117T substitution, wherein the substitution is positioned in accordance with the amino acid positions set forth in SEQ ID No. 1.

4. The method of claim 1 , wherein the chronic wound is a venous leg ulcer, venous foot ulcer, arterial leg ulcer, arterial foot ulcer, decubitus ulcer, pressure lesion, bedsore lesion, post-surgical ulcerous lesion, or a burn.

5. The method of claim 1 , wherein said subject is a diabetic.

6. The method of claim 1 , further comprising evaluating the healing process of said chronic wound.

7. The method of claim 1 , further comprising administering a local anesthetic agent to said subject.

8. The method of claim 1 , further comprising administering one or more antibacterial or antifungal agents to said subject.

9. The method of claim 1 , wherein said composition comprises 50 μg/g of said GM-CSF.

10. The method of claim 1 , wherein said composition comprises 80 μg/g to 120 μg/g of said GM-CSF.

11. The method of claim 1 , wherein said composition comprises 8-15% w/w of sucralfate.

12. The method of claim 1 , wherein said composition comprises 20% w/w of sucralfate.

13. The method of claim 1 , wherein said composition comprises 0.2-1.2% w/w of the salt of hyaluronan.

14. The method of claim 1 , wherein said composition comprises 0.2% w/w of the salt of hyaluronan.

15. The method of claim 1 , wherein said composition is formulated as a paste.

16. The method of claim 1 , wherein said composition provides moisture to the chronic wound.

17. The method of claim 16 , wherein the moisture facilitates alleviation to said chronic wound.

18. The method of claim 1 , wherein the chronic wound is a venous leg ulcer, venous foot ulcer, diabetic leg ulcer, diabetic foot ulcer, arterial leg ulcer, arterial foot ulcer, decubitus ulcer, pressure lesion, bedsore lesion, post-surgical ulcerous lesion, or a burn.

19. The method of claim 1 , wherein the salt of hyaluronan comprises a sodium salt, a potassium salt, a magnesium salt, a calcium salt, or a combination thereof.

20. The method of claim 1 , wherein the salt of hyaluronan comprises a sodium salt.

21. The method of claim 1 , wherein said GM-CSF is formulated in a liposome.

Assignments (2)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Apr 10, 2024
From: HESLET, LARS
To: TRIFOILIUM APS
Reel/Frame 067061/0976 →
CHANGE OF NAME Recorded Apr 10, 2024
From: TRIFOILIUM APS
To: REPONEX PHARMACEUTICALS A/S
Reel/Frame 067663/0277 →
Priority Claims (1)
DK PA 2014 70300 · May 23, 2014 · national
Continuity (2)
Continuation 15313384
Related Publication 20200030410A1 · Jan 30, 2020