IP Library Granted Patent US 12,504,430
Granted Patent B2
US 12,504,430 · App. 16/484,177 · Granted Dec 23, 2025

Methods for the detection and treatment of lung cancer

Inventors: Samir Hanash (Houston, TX); Ayumu Taguchi (Houston, TX); Ziding Feng (Houston, TX)
Assignee: Board of Regents, The University of Texas System
G01N33/57423G01N33/57484G16B5/20
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Quick Facts
Patent No.
US 12,504,430
App. No.
16/484,177
Granted
Dec 23, 2025
Kind
B2
Abstract

Provided are methods and related kits for detection of early stage lung cancer, and determination of risk of harboring lung cancer.

Claims (31)

1 . A method of determining the risk of a subject for harboring lung cancer and treating lung cancer, comprising

(a) measuring a level of biomarkers in a biological sample obtained from the subject, wherein the biomarkers comprise diacetylspermine (DAS), CEA, CA125, CYFRA21-1, and Pro-SFTPB, and wherein the biological sample is collected prior to a diagnosis of lung cancer;

(b) combining the measured levels into a biomarker-based risk score, wherein the biomarker-based risk score is calculated using logistic regression analysis and wherein the subject's biomarker-based risk score is elevated relative to a healthy subject;

(c) administering a computerized tomography (CT) scan or other imaging modality to the subject having the elevated biomarker-based risk score;

(d) classifying the subject as lung cancer positive based on the increased risk of having lung cancer quantified in step (b) and the imaging results obtained in step (c); and

(e) administering to the lung cancer positive subject a therapeutically effective amount of a treatment for the lung cancer comprising surgery, chemotherapy, immunotherapy, radiation therapy, targeted therapy, or a combination thereof.

2 . The method of claim 1 , wherein the lung cancer is non-small cell lung cancer, adenocarcinoma or squamous cell cancer.

3 . The method of claim 1 , wherein the lung cancer is diagnosed at or before the borderline resectable stage or at the resectable stage.

4 . The method of claim 1 , wherein the biological sample is selected from blood, plasma, and serum.

5 . The method of claim 1 , wherein the measuring of CEA, CA125, CYFRA21-1, pro-SFTPB, and DAS levels is made at substantially the same time or in a stepwise manner.

6 . The method of claim 1 , wherein measuring the level of biomarkers of CEA, CA125, CYFRA21-1, pro-SFTPB, and DAS comprises the use of one or more reporter molecules; and/or one or more surfaces capable of binding one or more biomarkers; and/or one or more relay molecules capable of binding one or more biomarkers.

7 . The method of claim 6 , wherein at least one of the surfaces is the surface of a solid particle.

8 . The method of claim 7 , wherein the solid particle is a bead.

9 . The method as recited in claim 6 , wherein at least one of the reporter molecules is linked to an enzyme, or wherein at least one of the reporter molecules provides a detectable signal.

10 . The method as recited in claim 9 , wherein the detectable signal is detectable by a method selected from UV-visible spectroscopy, mass spectrometry, nuclear magnetic resonance (NMR) spectroscopy, proton NMR spectroscopy, nuclear magnetic resonance (NMR) spectrometry, gas chromatography-mass spectrometry (GC-MS), liquid chromatography-mass spectrometry (LC-MS), correlation spectroscopy (COSy), nuclear Overhauser effect spectroscopy (NOESY), rotating frame nuclear Overhauser effect spectroscopy (ROESY), LC-TOF-MS, LC-MS/MS, and capillary electrophoresis-mass spectrometry.

11 . A method of treating a subject suspected of harboring lung cancer, comprising

(a) analyzing the subject for risk of harboring lung cancer with a method comprising:

(b) measuring a level of biomarkers in a biological sample obtained from the subject, wherein the biomarkers comprise diacetylspermine (DAS), CEA, CA125, CYFRA21-1, and Pro-SFTPB, and wherein the biological sample is collected prior to a diagnosis of lung cancer;

(c) combining the measured levels into a biomarker-based risk score, wherein the biomarker-based risk score is calculated using logistic regression analysis and wherein the biomarker-based risk score classifies the subject as being at risk of harboring lung cancer when the biomarker-based risk score is elevated in the subject relative to a healthy subject;

(d) classifying the subject as lung cancer positive based on the increased risk of having lung cancer quantified in step (c); and

(e) administering to the lung cancer positive subject a therapeutically effective amount of a treatment for the cancer.

12 . The method of treating of claim 11 , wherein the treatment is surgery, chemotherapy, immunotherapy, radiation therapy, targeted therapy, or a combination thereof.

13 . The method of claim 11 , wherein the lung cancer is adenocarcinoma or squamous cell cancer.

14 . The method of claim 11 , wherein the lung cancer is diagnosed at or before the borderline resectable stage or at the resectable stage.

15 . The method of claim 11 , wherein the biological sample is selected from blood, plasma, and serum.

16 . The method of claim 11 , wherein the measuring of CEA, CA125, CYFRA21-1, pro-SFTPB, and DAS levels is made at substantially the same time or in a stepwise manner.

17 . The method of claim 11 , wherein measuring the level of biomarkers of CEA, CA125, CYFRA21-1, pro-SFTPB, and DAS comprises the use of one or more reporter molecules; and/or one or more surfaces capable of binding one or more biomarkers; and/or one or more relay molecules capable of binding one or more biomarkers.

18 . The method of claim 17 , wherein at least one of the surfaces is the surface of a solid particle.

19 . The method as recited in claim 18 , wherein the solid particle is a bead.

20 . The method as recited in claim 17 , wherein at least one of the reporter molecules is linked to an enzyme; or wherein at least one of the reporter molecules provides a detectable signal.

21 . The method as recited in claim 20 , wherein the detectable signal is detectable by a method selected from UV-visible spectroscopy, mass spectrometry, nuclear magnetic resonance (NMR) spectroscopy, proton NMR spectroscopy, nuclear magnetic resonance (NMR) spectrometry, gas chromatography-mass spectrometry (GC-MS), liquid chromatography-mass spectrometry (LC-MS), correlation spectroscopy (COSy), nuclear Overhauser effect spectroscopy (NOESY), rotating frame nuclear Overhauser effect spectroscopy (ROESY), LC-TOF-MS, LC-MS/MS, and capillary electrophoresis-mass spectrometry.

Assignments (2)
CONFIRMATORY LICENSE Recorded Jun 17, 2020
From: UNIVERSITY OF TEXAS MD ANDERSON CANCER CENTER
To: THE GOVERNMENT OF THE UNITED STATES, AS REPRESENTED BY THE SECRETARY OF THE ARMY
Reel/Frame 052960/0566 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Aug 8, 2019
From: HANASH, SAMIR; TAGUCHI, AYUMU; FENG, ZIDING
To: BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM
Reel/Frame 050004/0591 →
Continuity (2)
Provisional Application 62456731 · Feb 9, 2017
Related Publication 20200025766A1 · Jan 23, 2020
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