IP Library Granted Patent US 10,835,512
Granted Patent B2
US 10,835,512 · App. 16/507,889 · Granted Nov 17, 2020

Methods of treating respiratory syncytial virus infections

Inventors: Pravin Soni (Sunnyvale, CA); William Gerhart (Del Mar, CA); Manfred Keller (Munich, DE); Ahmet Tutuncu (Del Mar, CA)
Assignee: Respivant Sciences GmbH
A61K31/352A61K9/0073A61K9/0075A61K9/0078A61K9/08A61K9/12A61K47/02
View Patent ↗
Loading inventors, assignments & file history…
Monitor This Case
Get email alerts when status or documents change.
Order Certified Copies
Most orders are placed with the USPTO same day — all within 24 business hours.
Order via The Patent Place →
Pre-filled with this patent's details
Quick Facts
Patent No.
US 10,835,512
App. No.
16/507,889
Granted
Nov 17, 2020
Kind
B2
Abstract

Compositions and methods for the treatment of respiratory syncytial virus infections are provided.

Claims (21)

1. A pharmaceutically acceptable aerosol for the treatment of a lung condition in a subject, consisting of droplets of a solution consisting of (i) from about 4% to about 6% by weight of cromolyn sodium and (ii) an osmolarity adjusting agent consisting of (a) between 0.1% and 0.5% by weight of sodium chloride, inclusive of the endpoints, and (b) optionally salts of ethylenediaminetetraacetic acid (EDTA), and (iii) water; wherein the aerosol has a respirable fraction (≤3.3 μm) as measured by USP <1601> of between about 30% and about 95%, inclusive of the endpoints, and wherein the treatment of the lung condition in the subject is achieved via delivery of a therapeutically effective amount of cromolyn sodium to the lungs of the subject by the subject orally inhaling the pharmaceutically acceptable aerosol.

2. The pharmaceutically acceptable aerosol of claim 1 , wherein the salts of EDTA comprise sodium EDTA.

3. The pharmaceutically acceptable aerosol of claim 1 , wherein the solution contains from about 5 mg to about 80 mg of cromolyn sodium.

4. The pharmaceutically acceptable aerosol of claim 1 , wherein the solution contains from about 36 mg to about 44 mg of cromolyn sodium.

5. The pharmaceutically acceptable aerosol of claim 1 , wherein the aerosol has a respirable fraction (≤5 μm) as measured by USP <1601> of between about 75% and about 95%, inclusive of the endpoints.

6. The pharmaceutically acceptable aerosol of claim 1 , wherein the sodium chloride is at a concentration of between 0.1% to 0.2% by weight, inclusive of the endpoints.

7. A pharmaceutically acceptable aerosol for delivery of a therapeutically effective amount of cromolyn sodium to the lungs of a subject, wherein the pharmaceutically acceptable aerosol is a nebulized solution consisting of (i) from about 4% to about 6% by weight of cromolyn sodium, (ii) between 0.1% and 0.5% by weight of sodium chloride, inclusive of the endpoints, (iii) a salt of EDTA, and (iv) water, wherein the delivery of a therapeutically effective amount of cromolyn sodium to the lungs of the subject is achieved by the subject orally inhaling the pharmaceutically acceptable aerosol.

8. The pharmaceutically acceptable aerosol of claim 7 , wherein the salt of EDTA is sodium EDTA.

9. The pharmaceutically acceptable aerosol of claim 7 , wherein the solution contains from about 5 mg to about 80 mg of cromolyn sodium.

10. The pharmaceutically acceptable aerosol of claim 7 , wherein the solution contains from about 36 mg to about 44 mg of cromolyn sodium.

11. The pharmaceutically acceptable aerosol of claim 7 , wherein the aerosol has a respirable fraction (≤3.3 μm) as measured by USP <1601> of between about 30% and about 95%, inclusive of the endpoints.

12. The pharmaceutically acceptable aerosol of claim 7 , wherein the aerosol has a respirable fraction (≤3.3 μm) as measured by USP <1601> of between about 30% and about 95%, inclusive of the endpoints, and a respirable fraction (≤5 μm) as measured by USP <1601> of between about 75% and about 95%, inclusive of the endpoints.

13. The pharmaceutically acceptable aerosol of claim 7 , wherein the sodium chloride is at a concentration of between 0.1% to 0.2% by weight, inclusive of the endpoints.

14. A method of treating a lung condition in a subject, comprising administering a pharmaceutically acceptable aerosol to the subject by oral inhalation, the pharmaceutically acceptable aerosol consisting of droplets of a solution consisting of (i) from about 4% to about 6% by weight of cromolyn sodium, (ii) between 0.1% and 0.5% by weight of sodium chloride, inclusive of the endpoints, (iii) optionally salts of ethylenediaminetetraacetic acid (EDTA), and (iv) water; wherein the aerosol has a respirable fraction (≤3.3 μm) as measured by USP <1601> of between about 30% and about 95%, inclusive of the endpoints.

15. The method of claim 14 , wherein the salts of EDTA comprise sodium EDTA.

16. The method of claim 14 , wherein the solution contains from about 5 mg to about 80 mg of cromolyn sodium.

17. The method of claim 14 , wherein the solution contains about from about 36 mg to about 44 mg of cromolyn sodium.

18. The method of claim 14 , wherein the aerosol has a respirable fraction (≤3.3 μm) as measured by USP <1601> of between about 30% and about 95%, inclusive of the endpoints.

19. The method of claim 14 , wherein the aerosol has a respirable fraction (≤5 μm) as measured by USP <1601> of between about 75% and about 95%, inclusive of the endpoints.

20. The method of claim 16 , wherein the aerosol has a further respirable fraction (≤5 μm) as measured by USP <1601> of between about 75% and about 95%, inclusive of the endpoints.

21. The method of claim 14 , wherein the sodium chloride is at a concentration of between 0.1% to 0.2% by weight, inclusive of the endpoints.

Assignments (3)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jul 27, 2020
From: GERHART, WILLIAM; KELLER, MANFRED; TUTUNCU, AHMET; SONI, PRAVIN
To: PATARA PHARMA, LLC
Reel/Frame 053319/0666 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jul 27, 2020
From: PATARA PHARMA, LLC
To: RESPIVANT SCIENCES LTD.
Reel/Frame 053319/0251 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jul 27, 2020
From: RESPIVANT SCIENCES LTD.
To: RESPIVANT SCIENCES GMBH
Reel/Frame 053319/0324 →
Continuity (7)
Continuation 15232747 · Aug 9, 2016
Continuation PCTUS2015015033 · Feb 9, 2015
Provisional Application 62105453 · Jan 20, 2015
Provisional Application 61978711 · Apr 11, 2014
Provisional Application 61971709 · Mar 28, 2014
Provisional Application 61937928 · Feb 10, 2014
Related Publication 20190328700A1 · Oct 31, 2019