IP Library Granted Patent US 11,078,535
Granted Patent B2
US 11,078,535 · App. 16/631,866 · Granted Aug 3, 2021

Presymptomatic micro RNA targets for treatment of neurodegeneration pathology

Inventors: Salil Sharma (Bloomington, IN); Hui-Chen Lu (Bloomington, IN)
Assignee: The Trustees of Indiana University
C12Q1/6883A61K31/7105A61P25/28C12N15/113C12Q1/686
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Quick Facts
Patent No.
US 11,078,535
App. No.
16/631,866
Granted
Aug 3, 2021
Kind
B2
Abstract

Compositions and methods are provided for the early detection of neuroinflammation in a patient in a presymptomatic stage of a neurodegenerative disease. The method comprises identifying patients with elevated expression levels of a micro RNA selected from the group consisting of miR142-3p, miR142-5p, miR181a, miR181b, miR219-3p and miR219-5p. The identified patients can then be treated with a therapeutic pharmaceutical composition comprising antimiR oligonucleotides.

Claims (12)

1. A method of treating neuroinflammation in a patient having a neurodegenerative condition and exhibiting elevated levels of two or more micro RNAs selected from the group consisting of miR142-3p, miR142-5p, and miR219-3p, said method comprising:

identifying in patients having a neurodegenerative condition, those patients having elevated levels of two or more micro RNAs selected from the group consisting of miR219-3p, miR142-3p and miR142-5, by

i) obtaining a reference expression level of two or more micro RNAs selected from the group consisting of miR219-3p, miR142-3p and miR142-5p;

ii) determining an expression level of two or more micro RNAs selected from the group consisting of miR219-3p, miR142-3p and miR142-5p, and corresponding to those of step i), in a sample obtained from said patient having a neurodegenerative condition, wherein an increase in the expression level of said two or more micro RNAs selected from the group consisting of miR142-3p and miR142-5p in said patient's sample as compared to the reference expression level identifies the patient as having neuroinflammation; and

administering to said patient having a neurodegenerative condition and identified as having elevated levels of said two or more micro RNAs selected from the group consisting of miR142-3p, miR142-5p, and miR219-3p a therapeutic composition comprising an antisense or interference oligonucleotide that is complementary to a micro RNA selected from the group consisting of miR142-3p, miR142-5p, and miR219-3p, wherein said antisense or interference oligonucleotide reduces the expression of a micro RNA selected from the group consisting of miR219-3p, miR142-3p and miR142-5p and provides treatment of said neuroinflammation.

2. A method of treating neuroinflammation in a patient with a neurodegenerative condition, said method comprising

i) obtaining a reference expression level of miR142-3p and miR219-3p;

ii) determining an expression level of miR142-3p and miR219-3p, in a sample obtained from said patient, wherein an increase in the expression level of miR142-3p and miR219-3p in said patient's sample as compared to the reference expression level identifies the patient as having neuroinflammation; and

administering a therapeutic composition comprising antisense or interference oligonucleotides that are complementary to the sequence of miR142-3p and miR219-3p to reduce the expression of miR142-3p and miR219-3p and treat said neuroinflammation.

3. The method of claim 2 further comprising the steps of

iii) obtaining a reference expression level of a micro RNA selected from the group consisting of miR142-5p, miR181a, miR181b, and miR219-5p;

iv) determining an expression level of a micro RNA selected from the group consisting of miR142-5p, miR181a, miR181b, and miR219-5p, in said test patient's sample, wherein an increase in the expression level of one or more of miR142-5p, miR181a, miR181b, and miR219-5p in said test patient's sample as compared to the reference expression level, in addition to the detected increase in expression levels of miR142-3p and miR219-3p, identifies the patient as having neuroinflammation.

Assignments (2)
CONFIRMATORY LICENSE Recorded Feb 18, 2020
From: INDIANA UNIVERSITY
To: NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT
Reel/Frame 051961/0471 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jan 29, 2020
From: SHARMA, SALIL; LU, HUI-CHEN
To: THE TRUSTEES OF INDIANA UNIVERSITY
Reel/Frame 051649/0357 →
Continuity (4)
Provisional Application 62665888 · May 2, 2018
Provisional Application 62660030 · Apr 19, 2018
Provisional Application 62533870 · Jul 18, 2017
Related Publication 20200157627A1 · May 21, 2020