IP Library Granted Patent US 11,400,076
Granted Patent B2
US 11,400,076 · App. 16/753,209 · Granted Aug 2, 2022

Cancer stem cell inhibitor

Inventors: Hideyuki Saya (Shinjuku-ku, JP); Oltea Sampetrean (Shinjuku-ku, JP); Naoyoshi Koike (Shinjuku-ku, JP); Nobuo Kubota (Shinagawa-ku, JP)
Assignees: KEIO UNIVERSITY; Sun Pharma Japan Limited
A61K31/4168A61K45/06
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Quick Facts
Patent No.
US 11,400,076
App. No.
16/753,209
Granted
Aug 2, 2022
Kind
B2
Abstract

The object of the present invention is to provide a novel pharmaceutical for suppressing cancer stem cells. In the present invention, a mitochondria inhibitor comprising a 2-nitroimidazole derivative is applied to the cancer stem cell as an active ingredient.

Claims (12)

1. A method for suppressing a cancer stem cell, the method comprising:

contacting the cancer stem cell with a pharmaceutical comprising a 2-nitroimidazole derivative as an active ingredient,

wherein the cancer stem cell is glioma, melanoma, or sarcoma, and

wherein the 2-nitroimidazole derivative is doranidazole, misonidazole, or etanidazole.

2. The method according to claim 1 , wherein the cancer stem cell is derived from metastatic cancer.

3. The method according to claim 1 , wherein the pharmaceutical is contacted together with a cancer damaging means.

4. The method according to claim 3 , wherein the cancer damaging means is administration of a cancer chemotherapeutic agent or radiation.

5. The method according to claim 3 , wherein the pharmaceutical is suitable for pretreatment, concurrent treatment, or posttreatment of the cancer damaging means.

6. A method for suppressing growth of a cancer stem cell, the method comprising:

administering a 2-nitroimidazole derivative to a subject in need thereof,

wherein the cancer stem cell is glioma, melanoma, or sarcoma, and

wherein the 2-nitroimidazole derivative is doranidazole, misonidazole, or etanidazole.

Assignments (2)
MERGER Recorded Jun 13, 2022
From: POLA PHARMA, INC.
To: SUN PHARMA JAPAN LIMITED
Reel/Frame 060180/0820 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Apr 2, 2020
From: SAYA, HIDEYUKI; SAMPETREAN, OLTEA; KOIKE, NAOYOSHI; KUBOTA, NOBUO
To: KEIO UNIVERSITY; POLA PHARMA INC.
Reel/Frame 052298/0907 →
Continuity (3)
Provisional Application 62587195 · Nov 16, 2017
Provisional Application 62566695 · Oct 2, 2017
Related Publication 20200316027A1 · Oct 8, 2020