IP Library Granted Patent US 11,298,343
Granted Patent B2
US 11,298,343 · App. 16/758,986 · Granted Apr 12, 2022

Method for treating thalassemia

Inventors: Mitchell J. Weiss (Memphis, TN); Mondira Kundu (Memphis, TN); Christophe Lechauve (Bartlett, TN)
Assignee: ST. JUDE CHILDREN'S RESEARCH HOSPITAL
A61K31/436A61P7/06A61K45/06
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Quick Facts
Patent No.
US 11,298,343
App. No.
16/758,986
Granted
Apr 12, 2022
Kind
B2
Abstract

Methods for removing excess free α-globin in erythroid cells and treating a thalassemia using an agent that activates Unc-51 Like autophagy activating Kinase (ULK) are described.

Claims (7)

1. A method for removing excess free α-globin in reticulocytes or erythrocytes comprising contacting reticulocytes or erythrocytes with an effective amount of an agonist that directly activates Unc-51 Like autophagy activating Kinase (ULK), AMP-Activated Protein Kinase (AMPK), or Glycogen synthase kinase 3 (GSK3) thereby removing excess free α-globin in the reticulocytes or erythrocytes.

2. A method for removing excess free, insoluble α-globin in reticulocytes or erythrocytes comprising contacting reticulocytes or erythrocytes with an effective amount of an agent that activates Unc-51 Like autophagy activating Kinase (ULK) thereby removing excess free, insoluble α-globin in the reticulocytes or erythrocytes, wherein the agent inhibits Mechanistic Target Of Rapamycin (mTOR).

3. A method for treating a thalassemia comprising administering to a subject in need thereof an effective amount of an agonist that directly activates Unc-51 Like autophagy activating Kinase (ULK), AMP-Activated Protein Kinase (AMPK), or Glycogen synthase kinase 3 (GSK3) and stimulates ULK1-dependent autophagy thereby treating the subject's thalassemia.

4. A method for treating a thalassemia comprising administering to a subject in need thereof an effective amount of an agent that activates Unc-51 Like autophagy activating Kinase (ULK), wherein the agent inhibits Mechanistic Target Of Rapamycin (mTOR) and is not an ATP-competitive mTOR kinase inhibitor.

5. The method of claim 3 , wherein the thalassemia is β-thalassemia.

6. The method of claim 4 , wherein the thalassemia is β-thalassemia.

7. The method of claim 2 , wherein the agent that inhibits mTOR is not an ATP-competitive mTOR kinase inhibitor.

Assignments (3)
CONFIRMATORY LICENSE Recorded Aug 12, 2020
From: ST. JUDE CHILDREN'S RESEARCH HOSPITAL
To: NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT
Reel/Frame 053465/0877 →
CONFIRMATORY LICENSE Recorded Aug 12, 2020
From: ST. JUDE CHILDREN'S RESEARCH HOSPITAL
To: NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT
Reel/Frame 053466/0253 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Apr 24, 2020
From: WEISS, MITCHELL J.; KUNDU, MONDIRA; LECHAUVE, CHRISTOPHE
To: ST. JUDE CHILDREN'S RESEARCH HOSPITAL
Reel/Frame 052487/0676 →
Continuity (2)
Provisional Application 62578104 · Oct 27, 2017
Related Publication 20200345702A1 · Nov 5, 2020