IP Library Granted Patent US 12,064,448
Granted Patent B2
US 12,064,448 · App. 16/762,845 · Granted Aug 20, 2024

Methods for reducing bioavailability and absorption of ingested substances

Inventors: Philip Demokritou (Brookline, MA); Glen Deloid (Natick, MA); Kee Woei Ng (Singapore, SG); Say Chye Joachim Loo (Singapore, SG)
Assignees: Nanyang Technological University; President and Fellows of Harvard College
A61K31/717A61K9/146
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Quick Facts
Patent No.
US 12,064,448
App. No.
16/762,845
Granted
Aug 20, 2024
Kind
B2
Abstract

Methods for reducing at least one of the bioavailability and absorption of at least one of ingested fat, carbohydrates, and unwanted substances from foodstuff in a subject are disclosed. The methods described herein include administering an amount of a nanobiopolymer, or combinations of nanobiopolymers, sufficient to reduce at least one of the bioavailability and absorption of ingested fat, carbohydrates, and unwanted substances to a subject, such as a human subject.

Claims (16)

1. A method for reducing the bioavailability and/or absorption of ingested fat from foodstuff in a subject, the method comprising:

administering an amount of a suspension of a nanobiopolymer, or combinations of nanobiopolymers, sufficient to reduce the bioavailability ingested fat to a subject,

wherein the nanobiopolymer is selected from the group consisting of cellulose nanofibers or cellulose nanocrystals and combinations thereof,

wherein, when the nanobiopolymer is cellulose nanofibers, the nanobiopolymer comprises fibrillar nanocellulose made by mechanical milling and having a diameter of up to 100 nm,

wherein when the nanobiopolymer is cellulose nanocrystals, the cellulose nanocrystals comprise nanocrystalline cellulose made by chemical means and the nanocrystalline cellulose ranges in diameter from 1 nm to 250 nm and

further wherein the bioavailability of the ingested fat is reduced by at least 30%.

2. The method of claim 1 , wherein the nanobiopolymer is incorporated into the foodstuff;

is administered separately from the foodstuff;

or is incorporated into the foodstuff and is administered separately from the foodstuff.

3. The method of claim 1 , wherein the amount of a nanobiopolymer sufficient to reduce the bioavailability and/or absorption of ingested fat from foodstuff is from about 0.75% to about 1.5% by weight of the foodstuff.

4. The method of claim 1 , wherein the fat comprises triglycerides.

5. The method of claim 1 , wherein the bioavailability and/or absorption of ingested fat is reduced by a reduction in translocation, in the subject's intestinal epithelium, of free fatty acids from triglycerides.

6. The method of claim 1 , wherein the bioavailability and/or absorption of ingested fat is reduced by modulating pancreatic lipase activity.

7. The method of claim 1 , wherein the bioavailability and/or absorption of ingested fat is reduced by inhibiting the hydrolysis of triglycerides.

8. The method of claim 1 , wherein the subject is a human subject.

9. The method of claim 1 , wherein the bioavailability of the ingested fat is reduced by at least 50%.

Assignments (3)
CONFIRMATORY LICENSE Recorded Oct 2, 2023
From: HARVARD UNIVERSITY
To: NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT
Reel/Frame 065090/0610 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Oct 8, 2020
From: DELOID, GLEN; DEMOKRITOU, PHILIP
To: PRESIDENT AND FELLOWS OF HARVARD COLLEGE
Reel/Frame 054012/0868 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Oct 8, 2020
From: LOO, SAY CHYE JOACHEM; NG, KEE WOEI
To: NANYANG TECHNOLOGICAL UNIVERSITY
Reel/Frame 054012/0917 →
Continuity (3)
Provisional Application 62697827 · Jul 13, 2018
Provisional Application 62584504 · Nov 10, 2017
Related Publication 20210030782A1 · Feb 4, 2021