IP Library Granted Patent US 11,376,253
Granted Patent B2
US 11,376,253 · App. 16/768,972 · Granted Jul 5, 2022

Agent for treating nocturnal pollakiuria

Inventors: Katsuya Segawa (Tokyo, JP); Takafumi Kurose (Tokyo, JP)
Assignee: KYORIN PHARMACEUTICAL CO., LTD.
A61K31/519A61P13/10A61K9/0053
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Quick Facts
Patent No.
US 11,376,253
App. No.
16/768,972
Granted
Jul 5, 2022
Kind
B2
Abstract

[Problem] To provide a novel therapeutic agent for nocturnal pollakiuria. [Solution] A therapeutic agent for nocturnal pollakiuria which contains, as an active ingredient, (6S)—N-[4-({(2S,5R)-5-[(R)-hydroxy(phenyl)methyl]pyrrolidin-2-yl}methyl)phenyl]-4-oxo-4,6,7,8-tetrahydropyrrolo[1,2-a]pyrimidine-6-carboxamide.

Claims (5)

1. A method for treating nocturnal pollakiuria, comprising administering to a subject in need thereof (6S)—N-[4-({(2S,5R)-5-[(R)-hydroxy(phenyl)methyl]pyrrolidin-2-yl}methyl)phenyl]-4-oxo-4,6,7,8-tetrahydropyrrolo[1,2-a]pyrimidine-6-carboxamide in an effective amount to treat nocturnal pollakiuria,

wherein the effective amount of the (6S)—N-[4-({(2S,5R)-5-[(R)-hydroxy(phenyl)methyl]pyrrolidin-2-yl}methyl)phenyl]-4-oxo-4,6,7,8-tetrahydropyrrolo[1,2-a]pyrimidine-6-carboxamide is administered to a subject belonging to a group of patients with nocturnal pollakiuria without nocturnal polyuria.

2. The method according to claim 1 , wherein the effective amount of the (6S)—N-[4-({(2S,5R)-5-[(R)-hydroxy(phenyl)methyl]pyrrolidin-2-yl}methyl)phenyl]-4-oxo-4,6,7,8-tetrahydropyrrolo[1,2-a]pyrimidine-6-carboxamide is administered to a subject belonging to a group of patients whose average value of the frequency of urination at night is 1.0 or more and 1.8 or less.

3. The method according to claim 1 , wherein the effective amount of the (6S)—N-[4-({(2S,5R)-5-[(R)-hydroxy(phenyl)methyl]pyrrolidin-2-yl}methyl)phenyl]-4-oxo-4,6,7,8-tetrahydropyrrolo[1,2-a]pyrimidine-6-carboxamide is administered orally once daily at a daily dosage of 50 mg or more and 100 mg or less.

4. The method according to claim 2 , wherein the effective amount of the (6S)—N-[4-({(2S,5R)-5-[(R)-hydroxy(phenyl)methyl]pyrrolidin-2-yl}methyl)phenyl]-4-oxo-4,6,7,8-tetrahydropyrrolo[1,2-a]pyrimidine-6-carboxamide is administered orally once daily at a daily dosage of 50 mg or more and 100 mg or less.

Assignments (4)
CHANGE OF ADDRESS Recorded Dec 25, 2024
From: KYORIN PHARMACEUTICAL CO., LTD.
To: KYORIN PHARMACEUTICAL CO., LTD.
Reel/Frame 069784/0473 →
MERGER Recorded Nov 13, 2023
From: KYORIN PHARMACEUTICAL CO., LTD.
To: KYORIN HOLDINGS, INC.
Reel/Frame 065545/0869 →
CHANGE OF NAME Recorded Nov 13, 2023
From: KYORIN HOLDINGS, INC.
To: KYORIN PHARMACEUTICAL CO., LTD.
Reel/Frame 065545/0960 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jun 2, 2020
From: SEGAWA, KATSUYA; KUROSE, TAKAFUMI
To: KYORIN PHARMACEUTICAL CO., LTD.
Reel/Frame 052809/0621 →
Priority Claims (2)
JP JP2017-244910 · Dec 21, 2017 · national
JP JP2018-212256 · Nov 12, 2018 · national
Continuity (1)
Related Publication 20210000831A1 · Jan 7, 2021