IP Library Granted Patent US 11,434,296
Granted Patent B2
US 11,434,296 · App. 16/798,030 · Granted Sep 6, 2022

Mitigation and reversal of intestinal fibrosis and inflammation by inhibition of TL1A function

Inventors: David Q. Shih (La Crescenta, CA); Stephan R. Targan (Santa Monica, CA); Dalin Li (Walnut, CA); Janine Bilsborough (Simi Valley, CA)
Assignee: CEDARS-SINAI MEDICAL CENTER
C07K16/2866A61K39/3955A61K45/06C07K16/24C07K16/241C07K16/2875C12N15/1138C12Q1/6883G01N33/6869C07K2317/76C12N2320/30C12Q2600/112C12Q2600/156C12Q2600/158G01N2333/7155G01N2800/065G01N2800/10
View Patent ↗
Loading inventors, assignments & file history…
Monitor This Case
Get email alerts when status or documents change.
Order Certified Copies
Most orders are placed with the USPTO same day — all within 24 business hours.
Order via The Patent Place →
Pre-filled with this patent's details
Quick Facts
Patent No.
US 11,434,296
App. No.
16/798,030
Granted
Sep 6, 2022
Kind
B2
Abstract

The invention relates to methods of treating fibrosis and inflammatory bowel disease. In one embodiment, the present invention treats gut inflammation by administering a therapeutically effective dosage of TL1A inhibitors and/or DR3 inhibitors to an individual. In another embodiment, the present invention provides a method of reversing tissue fibrosis in an individual by inhibiting TL1A-DR3 signaling function.

Claims (26)

1. A method of treating intestinal inflammation or fibrosis in a subject, comprising:

(a) determining whether a subject with intestinal inflammation or intestinal fibrosis has a high level of IL31RA relative to a level of IL31RA in a normal individual by:

(i) obtaining a sample from the subject; and

(ii) assaying the sample to detect a level of IL31RA; and

(b) if the level of IL31RA detected is high relative to a level of IL31RA in a normal individual, then administering to the subject a therapeutically effective dosage of an anti-TL1A antibody to treat the intestinal inflammation or intestinal fibrosis, wherein the anti-TL1A antibody is an inhibitor of TL1A-DR3 binding.

2. The method of claim 1 , wherein the subject has Crohn's disease or inflammatory bowel disease.

3. The method of claim 1 , wherein the subject has strictures in a small intestine.

4. The method of claim 1 , wherein the subject has intestinal fibrostenosis.

5. The method of claim 1 , wherein after administration, the level of IL31RA detected in the sample from the subject is reduced to a comparable level to the level of IL31RA in the normal individual.

6. A method of reversing intestinal fibrosis in a subject, comprising:

(a) determining whether a subject has intestinal fibrosis by:

(i) obtaining a sample from the subject; and

(ii) assaying the sample to detect a level of IL31RA; and

(b) reducing the number of intestinal primary fibroblasts in the subject by administering to the subject a therapeutically effective dosage of an anti-TL1A antibody, if the level of IL31RA detected is high relative to a level of IL31RA in a normal individual, wherein reducing the number of intestinal primary fibroblasts in the subject is effective to reverse intestinal fibrosis in the subject, wherein the anti-TL1A antibody is an inhibitor of TL1A-DR3 binding.

7. The method of claim 6 , wherein the subject has, or is suspected of having, an inflammatory bowel disease.

8. The method of claim 7 , wherein the inflammatory bowel disease is Crohn's disease.

9. The method of claim 6 , wherein the subject suffers from chronic inflammation.

10. The method of claim 6 , wherein the fibroblasts are myofibroblasts.

11. A method of reducing the number of intestinal primary fibroblasts in a subject, the method comprising:

(a) detecting in a sample obtained from a subject a high level of IL31RA relative to a level of IL31RA in a normal individual;

(b) administering to the subject from (a) an anti-TL1A antibody, thereby reducing the number of intestinal primary fibroblasts in the subject, wherein the anti-TL1A antibody is an inhibitor of TL1A-DR3 binding.

12. The method of claim 11 , wherein reducing the number of intestinal primary fibroblasts in the subject reduces the risk that the subject will develop intestinal fibrosis.

13. The method of claim 11 , wherein the subject has, or is suspected of having, an inflammatory bowel disease.

14. The method of claim 13 , wherein the inflammatory bowel disease is Crohn's disease.

15. The method of claim 11 , wherein the subject suffers from chronic inflammation.

16. The method of claim 11 , wherein the intestinal primary fibroblasts are myofibroblasts.

Assignments (1)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jul 20, 2020
From: SHIH, DAVID Q.; TARGAN, STEPHAN R.; LI, DALIN; BILSBOROUGH, JANINE
To: CEDARS-SINAI MEDICAL CENTER
Reel/Frame 053256/0409 →
Continuity (4)
Continuation 14779893
Provisional Application 61872020 · Aug 30, 2013
Provisional Application 61805806 · Mar 27, 2013
Related Publication 20200190203A1 · Jun 18, 2020
Cited By (5)
US 12,215,147 US 12,391,752 US 12,466,890 US 12,509,523 US 12,590,160