IP Library Granted Patent US 10,881,643
Granted Patent B2
US 10,881,643 · App. 16/842,814 · Granted Jan 5, 2021

Sphingosine pathway modulating compounds for the treatment of cancers

Inventors: Elazar Rabbani (New York, NY); James J. Donegan (Amesbury, MA)
Assignee: Enzo Biochem, Inc.
A61K31/4245A61K31/137A61P35/02
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Quick Facts
Patent No.
US 10,881,643
App. No.
16/842,814
Granted
Jan 5, 2021
Kind
B2
Abstract

The invention provides methods and compositions for treating cancers and myeloproliferative disorders using sphingosine kinase-1 inhibitors, such as SK1-I, and selective sphingosine-1-phosphate receptor agonists, such as ozanimod.

Claims (15)

1. A method for treating pancreatic cancer in a mammalian subject, comprising the step of:

coadministering to a mammalian subject in need of treatment for pancreatic cancer

(i) a therapeutically effective amount of ozanimod or a pharmaceutically acceptable salt thereof; and

(ii) a therapeutically effective amount of the compound

or a pharmaceutically acceptable salt thereof.

2. The method of claim 1 , wherein the mammalian subject is a human.

3. The method of claim 1 , wherein the coadministering step comprises:

coadministering to the mammalian subject the hydrochloride salt of the compound

4. The method of claim 3 , wherein the mammalian subject is a human.

5. The method of claim 1 , wherein the coadministering step comprises:

coadministering to the mammalian subject the hydrochloride salt of ozanimod.

6. The method of claim 5 , wherein the mammalian subject is a human.

7. The method of claim 3 , wherein the coadministering step comprises:

coadministering to the mammalian subject the hydrochloride salt of ozanimod.

8. The method of claim 7 , wherein the mammalian subject is a human.

Assignments (4)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jul 9, 2026
From: ENZO BIOCHEM, INC.; ENZO LIFE SCIENCES, INC.; ENZO THERAPEUTICS, INC.
To: SERAPH BIOTECH CONSULTING, LLC
Reel/Frame 075219/0465 →
RELEASE OF SECURITY INTEREST Recorded Jul 24, 2023
From: GEMINO HEALTHCARE FINANCE, LLC D/B/A SLR HEALTHCARE ABL
To: ENZO BIOCHEM, INC.; ENZO CLINICAL LABS, INC.; ENZO LIFE SCIENCES U.S. HOLDING CORP; ENZO LIFE SCIENCES, INC.
Reel/Frame 064369/0031 →
SECURITY INTEREST Recorded Apr 3, 2023
From: ENZO LIFE SCIENCES, INC.; ENZO CLINICAL LABS, INC.; ENZO BIOCHEM, INC.; ENZO LIFE SCIENCES U.S. HOLDING CORP
To: GEMINO HEALTHCARE FINANCE, LLC D/B/A SLR HEALTHCARE ABL
Reel/Frame 063239/0103 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Apr 16, 2020
From: RABBANI, ELAZAR; DONEGAN, JAMES J.; DIAMOND, PAUL
To: ENZO BIOCHEM, INC.
Reel/Frame 052411/0241 →
Continuity (4)
Division 16229490 · Dec 21, 2018
Continuation In Part 16017303 · Jun 25, 2018
Provisional Application 62524221 · Jun 23, 2017
Related Publication 20200230113A1 · Jul 23, 2020