IP Library Granted Patent US 11,160,796
Granted Patent B2
US 11,160,796 · App. 16/885,570 · Granted Nov 2, 2021

Anti-androgens for the treatment of non-metastatic castration-resistant prostate cancer

Inventor: Arturo Molina (Los Altos Hills, CA)
Assignee: Aragon Pharmaceuticals, Inc.
A61K31/4439A61K9/0053A61K31/00A61K31/192A61K31/4152A61K31/4155A61K31/4166A61K31/4178A61K31/426A61K31/427A61K31/4365A61K31/496A61P35/00G06Q30/0607
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Quick Facts
Patent No.
US 11,160,796
App. No.
16/885,570
Granted
Nov 2, 2021
Kind
B2
Abstract

Described herein are methods of treating non-metastatic castrate-resistant prostate cancer using an approved drug product comprising apalutamide, enzalutamide or darolutamide. Also described here are drug products containing apalutamide enzalutamide or darolutamide, and methods of selling or offering for sale an anti-androgen drug product.

Claims (11)

1. A method of improving metastasis free survival in a male human with non-metastatic castration-resistant prostate cancer, said method comprising administering to said male human an approved drug product comprising darolutamide in combination with androgen deprivation therapy.

2. The method of claim 1 , wherein the androgen deprivation therapy consists of orchiectomy or gonadotropin-releasing hormone agonists or antagonists.

3. The method of claim 1 , wherein the approved drug product provides an increase in the metastasis-free survival of the male human relative to the mean survival rate of a population of male humans with non-metastatic castration-resistant prostate cancer, said population having been administered a placebo in combination with androgen deprivation therapy.

4. The method of claim 1 , wherein a drug product label for a reference listed drug for such approved drug product comprises metastasis free survival data.

5. The method of claim 1 , wherein a drug product label for a reference listed drug for such approved drug product includes instructions for treating non-metastatic castration resistant prostate cancer.

6. The method of claim 1 , further comprising selling such approved drug product, wherein a drug product label for a reference listed drug for such approved drug product includes instructions for treating non-metastatic castration resistant prostate cancer.

7. The method of claim 6 , wherein the drug product label comprises metastasis free survival data.

8. A method of improving metastasis free survival in a male human with non-metastatic castration-resistant prostate cancer, said method comprising providing to said male human an approved drug product comprising darolutamide in combination with androgen deprivation therapy.

9. The method of claim 8 , wherein the androgen deprivation therapy consists of orchiectomy or gonadotropin-releasing hormone agonists or antagonists.

10. The method of claim 8 , wherein a drug product label for a reference listed drug for such approved drug product comprises metastasis free survival data.

11. The method of claim 8 , wherein a drug product label for a reference listed drug for such approved drug product includes instructions for treating non-metastatic castration resistant prostate cancer.

Assignments (3)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded May 23, 2023
From: MOLINA, ARTURO
To: ARAGON PHARMACEUTICALS, INC.
Reel/Frame 063727/0995 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded May 23, 2023
From: YU, MARGARET
To: JANSSEN RESEARCH & DEVELOPMENT, LLC
Reel/Frame 063728/0315 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded May 23, 2023
From: JANSSEN RESEARCH & DEVELOPMENT, LLC
To: ARAGON PHARMACEUTICALS, INC.
Reel/Frame 063728/0510 →
Continuity (5)
Continuation 15967452 · Apr 30, 2018
Provisional Application 62630594 · Feb 14, 2018
Provisional Application 62617745 · Jan 16, 2018
Provisional Application 62572791 · Oct 16, 2017
Related Publication 20200360361A1 · Nov 19, 2020
Cited By (1)
US 50,642