IP Library Granted Patent US 11,331,292
Granted Patent B2
US 11,331,292 · App. 16/894,110 · Granted May 17, 2022

Methods of treatment of cholestatic diseases

Inventor: Remy Hanf (Lille, FR)
Assignee: Genfit
A61K31/192A61P1/16A61K9/0053A61K45/06
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Quick Facts
Patent No.
US 11,331,292
App. No.
16/894,110
Granted
May 17, 2022
Kind
B2
Abstract

The present invention relates to the use of compound 1-[4-methylthiophenyl]-3-[3,5-dimethyl-4-carboxydimethylmethyloxyphenyl]prop-2-en-1-one (Elafibranor or GFT505) for treating cholestatic diseases, and more specifically PBC and/or PSC.

Claims (11)

1. A method for the treatment of primary biliary cholangitis, the method comprising orally administering elafibranor at a dose between 70 mg and 130 mg per administration to a subject with primary biliary cholangitis.

2. The method according to claim 1 , wherein the subject is a patient with primary biliary cholangitis and inadequate response to ursodeoxycholic acid.

3. The method according to claim 1 , the method comprising orally administering once daily 80 or 120 mg/day of elafibranor.

4. The method according to claim 1 , the method comprising orally administering once daily 80 mg/day of elafibranor.

5. The method according to claim 1 , the method further comprising administering to the subject another anti-cholestatic agent.

6. A method for the treatment of primary biliary cholangitis, comprising orally administering elafibranor at a dose between 70 mg and 130 mg per administration in combination with ursodeoxycholic acid to a subject with primary biliary cholangitis and inadequate response to ursodeoxycholic acid.

7. The method according to claim 6 , wherein elafibranor is administered at a dose of 80 mg per administration.

8. The method according to claim 6 , wherein elafibranor is orally administered once daily at a dose of 80 mg/day.

9. The method according to claim 6 , wherein elafibranor is administered at a dose of 120 mg per administration.

10. The method according to claim 6 , wherein elafibranor is orally administered once daily at a dose of 120 mg/day.

11. A method for the treatment of primary biliary cholangitis, comprising orally administering 80 mg/day of elafibranor once daily in combination with ursodeoxycholic acid to a subject with primary biliary cholangitis and inadequate response to ursodeoxycholic acid.

Assignments (1)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Oct 7, 2020
From: HANF, REMY
To: GENFIT
Reel/Frame 053994/0292 →
Priority Claims (1)
EP 16305381 · Mar 31, 2016 · regional
Continuity (2)
Continuation In Part 16090415
Related Publication 20200297672A1 · Sep 24, 2020
Cited By (7)
US 12,233,038 US 12,290,498 US 12,295,927 US 12,295,928 US 12,303,480 US 12,310,935 US 12,589,086