IP Library Granted Patent US 11,795,220
Granted Patent B2
US 11,795,220 · App. 16/904,510 · Granted Oct 24, 2023

Anti-PVRIG antibodies and methods of use

Inventors: Mark White (Antioch, CA); Sandeep Kumar (San Bruno, CA); Christopher Chan (South San Francisco, CA); Spencer Liang (San Mateo, CA); Lance Stapleton (Oakland, CA); Andrew W. Drake (Mountain View, CA); Yosi Gozlan (Tel Aviv, IL); Ilan Vaknin (Tel Aviv, IL); Shirley Sameah-Greenwald (Kfar Saba, IL); Liat Dassa (Tel Aviv, IL); Zohar Tiran (Oranit, IL); Gad S. Cojocaru (Tel Aviv, IL); Leonard Presta (San Francisco, CA); Richard Theolis (Santa Cruz, CA)
Assignee: COMPUGEN LTD.
C07K16/2803C07K7/06G01N33/57484C07K2317/21C07K2317/33C07K2317/34C07K2317/53C07K2317/55C07K2317/56C07K2317/565C07K2317/70C07K2317/74C07K2317/76C07K2317/92C07K2319/30C07K2319/32C12N15/1138C12N2310/14G01N2333/47
View Patent ↗
Loading inventors, assignments & file history…
Monitor This Case
Get email alerts when status or documents change.
Order Certified Copies
Most orders are placed with the USPTO same day — all within 24 business hours.
Order via The Patent Place →
Pre-filled with this patent's details
Quick Facts
Patent No.
US 11,795,220
App. No.
16/904,510
Granted
Oct 24, 2023
Kind
B2
Abstract

The present invention is directed to anti-PVRIG antibodies and methods of using same.

Claims (47)

1. A method of activating T-cells of a patient with cancer comprising administering an anti-PD-L1 antibody and an anti-PVRIG antibody to said patient, wherein said anti-PVRIG antibody comprises:

i) a heavy chain variable domain comprising the vhCDR1, vhCDR2, and vhCDR3 from SEQ ID NO:1434 and

ii) a light chain variable domain comprising the vlCDR1, vlCDR2, and vlCDR3 from SEQ ID NO:1453,

wherein a subset of said T-cells of said patient are activated.

2. The method according to claim 1 wherein said anti-PVRIG antibody comprises the heavy chain variable domain of SEQ ID NO:1434 and the light chain variable domain of SEQ ID NO:1453.

3. The method according to claim 2 wherein said anti-PVRIG antibody comprises the CH1-hinge-CH2-CH3 region from IgG1, IgG2, IgG3, or IgG4, wherein said hinge region optionally comprises mutations.

4. The method according to claim 3 wherein said anti-PVRIG antibody comprises the CL region of human kappa 2 light chain.

5. The method according to claim 1 wherein said T-cells are cytotoxic T-cells (CTLs).

6. The method according to claim 1 wherein said T-cells are selected from the group consisting of CD4 + T-cells and CD8 + T-cells.

7. The method according to claim 1 wherein said activation is measured as an increase in interferon-γ production and/or an increase in cytokine secretion.

8. A method of activating T-cells of a patient with cancer comprising administering an anti-PD-L1 antibody and an anti-PVRIG antibody to said patient, wherein said anti-PVRIG antibody comprises:

i) a heavy chain variable domain comprising the vhCDR1, vhCDR2, and vhCDR3 from SEQ ID NO:1447 and

ii) a light chain variable domain comprising the vlCDR1, vlCDR2, and vlCDR3 from SEQ ID NO:1462,

wherein a subset of said T-cells of said patient are activated.

9. The method according to claim 8 wherein said anti-PVRIG antibody comprises the heavy chain variable domain of SEQ ID NO:1447 and the light chain variable domain of SEQ ID NO:1462.

10. The method according to claim 9 wherein said anti-PVRIG antibody comprises the CH1-hinge-CH2-CH3 region from IgG1, IgG2, IgG3, or IgG4, wherein said hinge region optionally comprises mutations.

11. The method according to claim 10 wherein said anti-PVRIG antibody comprises the CL region of human kappa 2 light chain.

12. The method according to claim 9 wherein said T-cells are cytotoxic T-cells (CTLs).

13. The method according to claim 9 wherein said T-cells are selected from the group consisting of CD4+ T-cells and CD8+ T-cells.

14. The method according to claim 9 wherein said activation is measured as an increase in interferon-γ production and/or an increase in cytokine secretion.

15. A method of activating T-cells of a patient with cancer comprising administering an anti-PD-L1 antibody and an anti-PVRIG antibody to said patient, wherein said anti-PVRIG antibody comprises:

a) a heavy chain variable domain comprising:

i) a vhCDR1 comprising SEQ ID NO:885;

ii) a vhCDR2 comprising SEQ ID NO:886;

iii) a vhCDR3 comprising SEQ ID NO:887; and

b) a light chain variable domain comprising:

i) a vlCDR1 comprising SEQ ID NO:889;

ii) a vlCDR2 comprising SEQ ID NO:890;

iii) a vlCDR3 comprising SEQ ID NO:891,

wherein a subset of said T-cells of said patient are activated.

16. The method according to claim 15 wherein said anti-PVRIG antibody comprises the CH1-hinge-CH2-CH3 region from IgG1, IgG2, IgG3, or IgG4, wherein said hinge region optionally comprises mutations.

17. The method according to claim 16 wherein said anti-PVRIG antibody comprises the CL region of human kappa 2 light chain.

18. The method according to claim 15 wherein said T-cells are cytotoxic T-cells (CTLs).

19. The method according to claim 15 wherein said T-cells are selected from the group consisting of CD4 + T-cells and CD8 + T-cells.

20. The method according to claim 15 wherein said activation is measured as an increase in interferon-γ production and/or an increase in cytokine secretion.

21. A method of activating T-cells of a patient with cancer comprising administering an anti-PD-L1 antibody and an anti-PVRIG antibody to said patient, wherein said anti-PVRIG antibody comprises:

a) a heavy chain comprising:

i) a VH-CH-hinge-CH2-CH3, wherein the VH is SEQ ID NO:1434 and wherein the CH1-hinge-CH2-CH3 region is from IgG4; and

b) a light chain comprising:

i) a VL-CL, wherein the VL is SEQ ID NO:1453 and wherein the CL region is from human kappa 2 light chain.

22. The method according to claim 21 wherein said hinge region optionally comprises mutations.

23. A method of activating T-cells of a patient with cancer comprising administering an anti-PD-L1 antibody and an anti-PVRIG antibody to said patient, wherein said anti-PVRIG antibody comprises:

a) a heavy chain comprising:

i) a VH-CH1-hinge-CH2-CH3, wherein the VH is SEQ ID NO:1447 and wherein the CH1-hinge-CH2-CH3 region is from IgG4; and

b) a light chain comprising:

i) a VL-CL, wherein the VL is SEQ ID NO:1462 and wherein the CL region is from human kappa 2 light chain.

24. The method according to claim 23 wherein said hinge region optionally comprises mutations.

Assignments (3)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Nov 9, 2022
From: WHITE, MARK; KUMAR, SANDEEP; CHAN, CHRISTOPHER; LIANG, SPENCER; STAPLETON, LANCE; DRAKE, ANDREW W; GOZLAN, YOSI; VAKNIN, ILAN; SAMEAH-GREENWALD, SHIRLEY; DASSA, LIAT; TIRAN, ZOHAR; COJOCARU, GAD S; PRESTA, LEONARD
To: COMPUGEN LTD.
Reel/Frame 061710/0886 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Nov 9, 2022
From: WHITE, MARK; KUMAR, SANDEEP; CHAN, CHRISTOPHER; LIANG, SPENCER; STAPLETON, LANCE; DRAKE, ANDREW W; THEOLIS, RICHARD
To: COMPUGEN USA, INC.
Reel/Frame 061711/0078 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Nov 9, 2022
From: COMPUGEN USA, INC.
To: COMPUGEN LTD.
Reel/Frame 061711/0149 →
Continuity (7)
Continuation 16748695 · Jan 21, 2020
Continuation 15277980 · Sep 27, 2016
Division 15048967 · Feb 19, 2016
Provisional Application 62235823 · Oct 1, 2015
Provisional Application 62141120 · Mar 31, 2015
Provisional Application 62118208 · Feb 19, 2015
Related Publication 20210188974A1 · Jun 24, 2021