IP Library Granted Patent US 12,090,142
Granted Patent B2
US 12,090,142 · App. 16/975,092 · Granted Sep 17, 2024

Combination therapy for the treatment of cancer

Inventors: Satish K. Srivastava (Galveston, TX); Kota V. Ramana (Galveston, TX); Ashish Saxena (Galveston, TX)
Assignee: Board of Regents, The University of Texas System
A61K31/4188A61K39/3955A61P35/00C07K16/2818A61K2039/505
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Quick Facts
Patent No.
US 12,090,142
App. No.
16/975,092
Granted
Sep 17, 2024
Kind
B2
Abstract

Certain embodiments are directed to methods and compositions for treating cancer, specifically colorectal cancer by administering an aldose reductase inhibitor and an immune checkpoint inhibitor to a subject in need thereof. Certain embodiments are directed to methods of treating a subject having cancer comprising, administering (i) a composition comprising an aldose reductase specific inhibitor and (ii) a composition comprising an immune checkpoint inhibitor to the subject having melanoma, head and neck, or colorectal cancer.

Claims (7)

1. A method of treating a subject having cancer comprising, administering (i) a composition comprising an aldose reductase specific inhibitor, wherein the aldose reductase specific inhibitor is fidarestat, and (ii) a composition comprising an immune checkpoint inhibitor, wherein the immune checkpoint inhibitor is anti-PD1, to the subject having cancer.

2. The method of claim 1 , wherein the cancer is melanoma, head and neck, bladder, breast, lung, or colorectal cancer.

3. The method of claim 1 , further comprising a second immune checkpoint inhibitor.

4. The method of claim 3 , wherein the second immune checkpoint inhibitor and the first immune checkpoint inhibitor inhibit different pathways.

5. The method of claim 1 , wherein the aldose reductase specific inhibitor is administered about 1, 2, 3, 4, 5, 6, 7, 8, 9, 10, hours or days prior to administration of the immune checkpoint inhibitor.

6. The method of claim 1 , wherein the cancer is premalignant, malignant, metastatic, or drug-resistant.

7. An anti-cancer composition comprising fidarestat and anti-PD1.

Assignments (2)
CONFIRMATORY LICENSE Recorded Oct 12, 2022
From: UNIVERSITY OF TEXAS MED BR GALVESTON
To: NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT
Reel/Frame 061656/0661 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Aug 24, 2020
From: SRIVASTAVA, SATISH K.; RAMANA, KOTA V.; SAXENA, ASHISH
To: THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM
Reel/Frame 053578/0054 →
Continuity (2)
Provisional Application 62633820 · Feb 22, 2018
Related Publication 20210085650A1 · Mar 25, 2021