IP Library Granted Patent US 12,221,489
Granted Patent B2
US 12,221,489 · App. 17/004,331 · Granted Feb 11, 2025

Antibodies to human B7x for treatment of metastatic cancer

Inventors: Xingxing Zang (New York, NY); James P. Allison (Houston, TX)
Assignees: ALBERT EINSTEIN COLLEGE OF MEDICINE; SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH
C07K16/30A61K9/0019A61K39/3955A61K39/39558A61K45/06A61K49/0008C07K16/28C07K16/2827C07K16/3015C07K16/3023C07K16/303C07K16/3038C07K16/3046C07K16/3053C07K16/3069G01N33/5011A61K2039/505C07K2317/34C07K2317/732C07K2317/76C07K2317/92
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Quick Facts
Patent No.
US 12,221,489
App. No.
17/004,331
Granted
Feb 11, 2025
Kind
B2
Abstract

Methods are provided for treating metastatic cancer in patients having metastatic cancer or for preventing metastasis in cancer patients at risk for metastasis comprising administering to the patient an antibody to B7x, or an active antibody fragment that binds B7x, in an amount effective to treat or prevent metastasis.

Claims (13)

1. An IgG1 monoclonal antibody or a fragment thereof comprising a means for selectively binding to human B7x amino acid residues 35-148 of SEQ ID NO: 1 with an equilibrium dissociation constant from residues 35-148 of SEQ ID NO: 1 that is less than 50 nM, wherein the IgG1 monoclonal antibody is capable of killing tumor cells through antibody-dependent cellular cytotoxicity.

2. The IgG1 monoclonal antibody or a fragment thereof of claim 1 , wherein the IgG1 monoclonal antibody or fragment blocks inhibition of T cell function by binding to B7x.

3. The IgG1 monoclonal antibody or a fragment thereof of claim 1 , wherein the IgG1 monoclonal antibody or fragment thereof does not include an antibody-partner molecule conjugate.

4. An IgG1 monoclonal antibody or a fragment thereof comprising a means for selectively binding to human B7x amino acid residues 35-148 of SEQ ID NO: 1 with an equilibrium dissociation constant from residues 35-148 of SEQ ID NO: 1 that is less than 50 nM, wherein the IgG1 monoclonal antibody is capable of preventing reoccurrence of a tumor by blocking inhibition of T cell function by B7x.

5. An IgG1 monoclonal antibody or a fragment thereof comprising a means for selectively binding to human B7x amino acid residues 35-148 of SEQ ID NO:1 with an equilibrium dissociation constant from residues 35-148 of SEQ ID NO: 1 that is less than 50 nM, wherein the IgG1 monoclonal antibody is capable of (i) treating a metastatic cancer or (ii) preventing metastasis of a cancer.

6. The IgG1 monoclonal antibody or a fragment thereof of claim 5 , wherein a first level of B7x expression in a tumor sample from the metastatic cancer or the cancer is determined, and the first level of B7x expression in the tumor sample-is compared to a second level of B7x expression in a corresponding healthy tissue.

7. The IgG1 monoclonal antibody or a fragment thereof of claim 5 , wherein the metastatic cancer or the cancer is a cancer of the skin, breast, pancreas, prostate, ovary, kidney, esophagus, gastrointestinal tract, colon, brain, liver, lung, head and/or neck.

8. A combination of anti-cancer agents comprising the IgG1 monoclonal antibody or a fragment thereof of claim 1 , and a second anti-cancer agent that is not bound to the IgG1 monoclonal antibody or a fragment thereof.

9. The combination of claim 8 , wherein the second anti-cancer agent is selected from the group consisting of an antibody against CTLA-4, an antibody against PD-1, an anti-EGFR agent, an alkylating agent, paclitaxel, docetaxel, and a topoisomerase inhibitor.

10. The combination of claim 9 , wherein the second anti-cancer agent is an antibody against CTLA-4.

11. The combination of claim 9 , wherein the anti-EGFR agent is selected from the group consisting of panitumumab, cetuximab, gefitinib and erlotinib.

12. The combination of claim 9 , wherein the alkylating agent is selected from the group consisting of cisplatin, carboplatin, oxaliplatin, nedaplatin, satraplatin, triplatin tetranitrate, mechlorethamine, cyclophosphamide, chlorambucil and ifosfamide.

13. The combination of claim 9 , wherein the topoisomerase inhibitor is selected from the group consisting of irinotecan, topotecan, amsacrine, etoposide, etoposide phosphate and teniposide.

Assignments (7)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Apr 22, 2024
From: ALLISON, JAMES P.
To: HOWARD HUGHES MEDICAL INSTITUTE
Reel/Frame 067183/0371 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Apr 22, 2024
From: HOWARD HUGHES MEDICAL INSTITUTE
To: SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH
Reel/Frame 067183/0432 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Apr 22, 2024
From: ZANG, XINGXING
To: ALBERT EINSTEIN COLLEGE OF MEDICINE OF YESHIVA UNIVERSITY
Reel/Frame 067183/0851 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Apr 22, 2024
From: ALBERT EINSTEIN COLLEGE OF MEDICINE OF YESHIVA UNIVERSITY
To: COM AFFILIATION, INC.
Reel/Frame 067184/0011 →
MERGER AND CHANGE OF NAME Recorded Apr 22, 2024
From: ALBERT EINSTEIN COLLEGE OF MEDICINE, INC.; ALBERT EINSTEIN COLLEGE OF MEDICINE
To: ALBERT EINSTEIN COLLEGE OF MEDICINE
Reel/Frame 067184/0101 →
EXECUTIVE ORDER 9424, CONFIRMATORY LICENSE Recorded Apr 22, 2024
From: YESHIVA UNIVERSITY
To: NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT
Reel/Frame 067187/0772 →
CHANGE OF NAME Recorded Apr 22, 2024
From: COM AFFILIATION, INC.
To: ALBERT EINSTEIN COLLEGE OF MEDICINE, INC.
Reel/Frame 067188/0220 →
Continuity (5)
Continuation 15252267 · Aug 31, 2016
Division 14050512 · Oct 10, 2013
Continuation In Part PCTUS2012034348 · Apr 20, 2012
Provisional Application 61477729 · Apr 21, 2011
Related Publication 20200392246A1 · Dec 17, 2020
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