IP Library Granted Patent US 11,725,023
Granted Patent B2
US 11,725,023 · App. 17/166,071 · Granted Aug 15, 2023

Therapeutic oligonucleotides

Inventors: Heather O'Neill (Mesa, AZ); Günter Mayer (Bonn, DE); Mark Miglarese (Phoenix, AZ); David Spetzler (Paradise Valley, AZ)
Assignee: Caris Science, Inc.
C07H19/173A61K9/0014A61K9/0019A61K9/0053A61K47/6911A61K47/6929A61P9/00A61P25/28A61P29/00A61P31/00A61P35/02A61P37/00C07H19/09C07H19/19C07H21/00C12N15/10C12N15/115C12Q1/6886G01N33/5308G01N33/57484G01N33/68G06T7/0012C12N2310/16C12N2320/10C12Q2600/158
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Quick Facts
Patent No.
US 11,725,023
App. No.
17/166,071
Granted
Aug 15, 2023
Kind
B2
Abstract

Methods and compositions are provided for oligonucleotides that bind targets of interest. The targets include cells and microvesicles, such as those derived from various diseases. The oligonucleotides can be used for diagnostic and therapeutic purposes. The target of the oligonucleotides can be a target such as PARP1, HIST1H1B, HIST1H1D, NCL, FBL, SFPQ, RPL12, ACTB, HIST1H4A, SSBP1, NONO, H2AFJ, and DDX21, or a complex, subunit or fragment thereof.

Claims (14)

1. An oligonucleotide consisting of SEQ ID NO. 4357.

2. A composition comprising an oligonucleotide consisting of SEQ ID NO. 4357.

3. A method comprising synthesizing the oligonucleotide according to claim 1 .

4. A method comprising contacting a biological sample with the oligonucleotide according to claim 1 .

5. The method of claim 4 , further comprising detecting a presence or level of a protein represented by a UniProt accession number selected from the group consisting of P19338, P22626, P06748, P60709, P22087, P09651, Q04837, P11142, Q00839, P52272, Q07955, P55769, Q12906, P06576, P31942, Q86V81, Q9NR30, Q96PK6, P37108, P09874, P17096, Q99729, P11021, P23246, P27694, Q13151, P04792, P31943, P51991, P02647, 043390, P08865, 014979, Q15365, P26599, Q14624, Q14103, P04406, 060506, Q15717, Q8NFH5, Q9NX24, P01009, Q14978, P10809, P14866, Q13243, Q6RFH5, Q9NZI8, P46087, P18754, P11940, P25705, Q15173, Q9Y3B9, Q9Y3Y2, P84103, P30154, Q00577, 1A31_HUMAN, 000479, P62263, Q16629, P52907, Q12905, P13645, P07910, Q7L8J4, P14923, P16403, P62633, P61978, P35268, Q01844, Q9UKM9, Q14978-1, P62750, P68431, P67809, P50914, Q8TEM1, P46087-4, Q13435, P23246-1, Q9NR30-1, P11387, Q14978-2, P17480-1, Q12906-7, Q9NVP1, Q13769, Q08170, P17844, P11940-1, 000567, P05109, Q15233, P06702, Q06830, P25311, P38159-1, P07910-1, P35678, Q05639, 060832-1, Q13601, Q15287-1, P61978-2, Q13247, P42696, Q969G3, P04406-1, P07910-2, Q9UKM9-1, P09651-1, Q08188, P07355-2, P16402, P16401, P62979, Q9BTM1, Q5D862, P30050-1, P31151, Q9NY12-1, P62633-1, P15927-3, P62913, P62081, P14678-3, Q9BRL6-1, Q92522, Q07020, P26373-1, Q92979, P09661, Q04387, P62805, P04908, Q5QNW6-2, P53999, P06899, P62888, P62899-2, P61353, P62318, P69905, Q8IUE6, P62829, P62851, P62269, P60866-2, and P49458 in the biological sample that is bound by the oligonucleotide.

6. The method of claim 4 , further comprising detecting a presence or level of a protein represented by a UniProt accession number selected from the group consisting of P09874, P16401, P16402, P19338, P22087, P23246, P30050, P60709, P628-5, Q04837, Q15233, Q9BTM1, and Q9NR30 in the biological sample that is bound by the oligonucleotide.

7. A pharmaceutical composition comprising a therapeutically effective amount of the oligonucleotide according to claim 1 , or a salt thereof, and a pharmaceutically acceptable carrier, diluent, or both.

8. The pharmaceutical composition of claim 7 , wherein the oligonucleotide is attached to a toxin or chemotherapeutic agent.

9. A method of modulating proliferation of a cell, comprising contacting the cell with the composition of claim 2 .

10. The method of claim 9 , wherein the composition induces apoptosis.

11. The method of claim 9 , wherein the cell is a leukemia cell, a lymphoma cell or a renal carcinoma cell.

12. The method of claim 9 , wherein the cell is a Ramos cell.

13. The method of claim 9 , wherein the cell expresses surface nucleolin.

14. The method of claim 9 , wherein the cell expresses heterogeneous nuclear ribonucleoprotein U protein (HNRPU) on its surface.

Assignments (4)
RELEASE OF SECURITY INTEREST IN PATENTS AT REEL/FRAME NO. 62419/0390 Recorded Apr 1, 2026
From: WILMINGTON TRUST, NATIONAL ASSOCIATION, AS ADMINISTRATIVE AGENT
To: CARIS MPI, INC.; CARIS SCIENCE, INC.
Reel/Frame 075424/0290 →
PATENT SECURITY AGREEMENT Recorded Apr 1, 2026
From: CARIS SCIENCE, INC.
To: BLUE OWL CAPITAL CORPORATION, AS ADMINISTRATIVE AGENT
Reel/Frame 075362/0668 →
SECURITY INTEREST Recorded Jan 18, 2023
From: CARIS MPI, INC.; CARIS SCIENCE, INC.
To: WILMINGTON TRUST, NATIONAL ASSOCIATION
Reel/Frame 062419/0390 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Feb 16, 2021
From: O'NEILL, HEATHER; MAYER, GÜNTER; MIGLARESE, MARK; SPETZLER, DAVID
To: CARIS SCIENCE, INC.
Reel/Frame 056859/0418 →
Continuity (8)
Continuation 15745407
Provisional Application 62305536 · Mar 9, 2016
Provisional Application 62269671 · Dec 18, 2015
Provisional Application 62239226 · Oct 8, 2015
Provisional Application 62220652 · Sep 18, 2015
Provisional Application 62198051 · Jul 28, 2015
Provisional Application 62198110 · Jul 28, 2015
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