IP Library Granted Patent US 11,555,025
Granted Patent B2
US 11,555,025 · App. 17/345,844 · Granted Jan 17, 2023

Crystalline form of N-[1-(5-cyano-pyridin-2-ylmethyl)-1 H-pyrazol-3-yl]-2- [4-(1-trifluoromethyl-cyclopropyl)-phenyl-acetamide

Inventors: Bibia Heidmann (Allschwil, CH); Markus Von Raumer (Allschwil, CH)
Assignee: IDORSIA PHARMACEUTICALS LTD
C07D401/06C07B2200/13
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Quick Facts
Patent No.
US 11,555,025
App. No.
17/345,844
Granted
Jan 17, 2023
Kind
B2
Abstract

The present invention relates to crystalline forms of N-[1-(5-cyano-pyridin-2-ylmethyl)-1H-pyrazol-3-yl]-2-[4-(1-trifluoromethyl-cyclopropyl)-phenyl]-acetamide, pharmaceutical compositions comprising said crystalline forms and their use as T-type calcium channel blockers in the treatment or prevention of diseases or disorders where T-type calcium channels are involved.

Claims (2)

1. A crystalline form of N-[1-(5-cyano-pyridin-2-ylmethyl)-1H-pyrazol-3-yl]-2-[4-(1-trifluoromethyl-cyclopropyl)-phenyl]-acetamide, characterized by the presence of an endothermic peak in the differential scanning calorimetry (DSC) thermogram at 147±2° C.

2. The crystalline form of claim 1 , wherein the crystalline form has peaks in the X-ray powder diffraction diagram at the following angles of refraction 2θ: 4.7°, 14.1°, and 20.1°.

Assignments (2)
PATENT SECURITY AGREEMENT Recorded Jun 25, 2026
From: IDORSIA PHARMACEUTICALS LTD
To: BIOPHARMA CREDIT PLC, AS COLLATERAL AGENT
Reel/Frame 076038/0461 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Aug 11, 2021
From: HEIDMANN, BIBIA; VON RAUMER, MARKUS
To: IDORSIA PHARMACEUTICALS LTD
Reel/Frame 057145/0992 →
Continuity (2)
Continuation 16628618
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