IP Library Granted Patent US 11,667,718
Granted Patent B2
US 11,667,718 · App. 17/359,986 · Granted Jun 6, 2023

Cancer treatment

Inventors: Mihael H. Polymeropoulos (Potomac, MD); Louis William Licamele (Potomac, MD); Christian Lavedan (Potomac, MD)
Assignee: Vanda Pharmaceuticals Inc.
C07K16/2866A61K9/0019A61K9/0053A61K9/0095A61K9/08A61K9/10A61K9/107A61K9/48A61K31/165A61K38/00A61K2039/505C07K2317/21C07K2317/565C07K2317/76
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Quick Facts
Patent No.
US 11,667,718
App. No.
17/359,986
Filed
Jun 28, 2021
Granted
Jun 6, 2023
Kind
B2
Art Unit
1623
USPC
424/172.1
Abstract

The invention relates generally to the treatment of cancer. One embodiment of the invention provides a method of treating cancer in an individual, the method comprising: administering to the individual an effective amount of trichostatin A (TSA).

Claims (13)

1. In a method of treating a patient diagnosed with cancer with trichostatin A (TSA), the improvement comprising:

selecting for treatment a patient determined to have increased aurora kinase A (AURKA) expression,

wherein the treating includes administering TSA to the selected patient in an amount sufficient to decrease an AURKA level in the selected patient.

2. The improvement of claim 1 , wherein the amount of TSA is sufficient to inhibit histone deacetylase (HDAC) activity in the selected patient.

3. The improvement of claim 1 , wherein the amount of TSA is between about 0.1 mg/kg/day and about 10 mg/kg/day.

4. The improvement of claim 3 , wherein the amount of TSA is between about 0.5 mg/kg/day and about 5 mg/kg/day.

5. The improvement of claim 1 , wherein the cancer is selected from a group consisting of: breast cancer, gastric cancer, colon cancer, rectal cancer, bladder cancer, pancreatic cancer, ovarian cancer, prostate cancer, lung cancer, hematological cancer, and skin cancer.

6. The improvement of claim 1 , wherein the TSA is administered orally.

7. The improvement of claim 1 , wherein the TSA is administered intravenously.

8. The improvement of claim 1 , further comprising:

determining, from a tumor sample obtained from the selected patient's body, a level of aurora kinase A (AURKA) expression.

9. The improvement of claim 1 , wherein the cancer is breast cancer.

10. The improvement of claim 1 , wherein the cancer is a malignancy.

Assignments (1)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jun 30, 2021
From: POLYMEROPOULOS, MIHAEL H.; LICAMELE, LOUIS WILLIAM; LAVEDAN, CHRISTIAN
To: VANDA PHARMACEUTICALS INC.
Reel/Frame 056718/0808 →
Continuity (5)
Continuation 16357249 · Mar 18, 2019
Continuation 15980644 · May 15, 2018
Continuation 14912077
Provisional Application 61869039 · Aug 22, 2013
Related Publication 20210324093A1 · Oct 21, 2021
Cited By (2)
US 12,590,162 US 12,673,033