IP Library Granted Patent US 12,577,282
Granted Patent B2
US 12,577,282 · App. 17/434,616 · Granted Mar 17, 2026

Galectin-1/ galectin-3 chimeras and multivalent proteins

Inventors: Gregory Allan Hudalla (Gainesville, FL); Margaret Mary Fettis (Northborough, MA)
Assignee: University of Florida Research Foundation, Incorporated
C07K14/4726A61P29/00A61K38/00C07K2319/73
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Quick Facts
Patent No.
US 12,577,282
App. No.
17/434,616
Granted
Mar 17, 2026
Kind
B2
Abstract

Described herein are Galectin-1/Galectin-3 multivalent protein complexes and uses thereof. In some aspects, Galectin-1/Galectin-3 multivalent protein complexes are useful to treat inflammatory conditions in a subject.

Claims (44)

1 . A Galectin-1/Galectin-3 (Gal-1/Gal-3) dimer comprising:

two monomer polypeptides, wherein each monomer polypeptide comprises:

a Galectin-1 (Gal-1) polypeptide;

a Galectin-3 (Gal-3) polypeptide; and

a linker comprising an alpha helix coil, wherein the alpha helix coil comprises the sequence of SEQ ID NO: 9, wherein the linker is fused between the Gal-1 polypeptide and the Gal-3 polypeptide,

wherein the two monomer polypeptides associate with each other via dimerization at the alpha helix coils to form the Gal-1/Gal-3 dimer, wherein one or both of the monomer polypeptides has a sequence that is about 90% to about 100% identical to SEQ ID NO: 3.

2 . The Gal-1/Gal-3 dimer of claim 1 , wherein the Gal-1 polypeptide has a sequence that is about 80% to about 100% identical to SEQ ID NO: 1.

3 . The Gal-1/Gal-3 dimer of claim 1 , wherein the Gal-3 polypeptide has a sequence that is about 80% to about 100% identical to SEQ ID NO: 4.

4 . The Gal-1/Gal-3 dimer of claim 1 , wherein the alpha helix coil has a sequence that is about 80% to about 100% identical to SEQ ID NO: 5.

5 . A pharmaceutical formulation comprising:

the Galectin-1/Galectin-3 (Gal-1/Gal-3) dimer of claim 1 ; and

a pharmaceutically acceptable carrier.

6 . A Galectin-1/Galectin-3 (Gal-1/Gal-3) polypeptide capable of dimerizing comprising:

a Galectin-1 (Gal-1) polypeptide;

a Galectin-3 (Gal-3) polypeptide; and

a linker comprising an alpha helix coil, wherein the alpha helix coil comprises the sequence of SEQ ID NO: 9, wherein the linker is fused between the Gal-1 polypeptide and the Gal-3 polypeptide, wherein the Gal-1/Gal-3 polypeptide has a sequence that is about 90% to about 100% identical to SEQ ID NO: 3.

7 . The Galectin-1/Galectin-3 (Gal-1/Gal-3) dimer of claim 1 , wherein:

(i) the Gal-1 polypeptide in at least one of the monomer polypeptides comprises the sequence of SEQ ID NO: 1;

(ii) the linker in at least one of the monomer polypeptides comprises the sequence of any one of SEQ ID NOs: 5, 10, or 11;

and/or

(iii) at least one of the monomer polypeptides does not comprise an N-terminal tag or a C-terminal tag.

8 . A pharmaceutical formulation comprising:

a plurality of the Galectin-1/Galectin-3 (Gal-1/Gal-3) polypeptide of claim 6 ; and

a pharmaceutically acceptable carrier.

9 . The Gal-1/Gal-3 polypeptide of claim 6 , wherein the Gal-1 polypeptide has a sequence that is about 80% to about 100% identical to SEQ ID NO: 1.

10 . The Gal-1/Gal-3 polypeptide of claim 6 , wherein the Gal-3 polypeptide has a sequence that is about 80% to about 100% identical to SEQ ID NO: 4.

11 . The Gal-1/Gal-3 polypeptide of claim 6 , wherein the alpha helix coil has a sequence that is about 80% to about 100% identical to SEQ ID NO: 5.

12 . The Galectin-1/Galectin-3 (Gal-1/Gal-3) polypeptide of claim 6 , wherein:

(i) the Gal-1 polypeptide comprises the sequence of SEQ ID NO: 1;

(ii) the linker comprises the sequence of any one of SEQ ID NOs: 5, 10, or 11;

and/or

(iii) the Gal-1/Gal-3 polypeptide does not comprise an N-terminal tag or a C-terminal tag.

13 . A Galectin-1/Galectin-3 (Gal-1/Gal-3) polynucleotide comprising:

a polynucleotide that encodes a Galectin-1 (Gal-1) polypeptide;

a polynucleotide that encodes a Galectin-3 (Gal-3) polypeptide; and

a polynucleotide that encodes a linker comprising an alpha helix coil, wherein the alpha helix coil comprises the sequence of SEQ ID NO: 9, wherein the polynucleotide that encodes the alpha helix coil is fused in-frame between the polynucleotide that encodes the Gal-1 polypeptide and the polynucleotide that encodes the Gal-3 polypeptide, wherein the Gal-1/Gal-3 polynucleotide encodes a polypeptide having a sequence that is about 90% to about 100% identical to SEQ ID NO: 3.

14 . The Gal-1/Gal-3 polynucleotide of claim 13 , wherein the Gal-1 polypeptide has a sequence that is about 80% to about 100% identical to SEQ ID NO: 1.

15 . The Gal-1/Gal-3 polynucleotide of claim 13 , wherein the Gal-3 polypeptide has a sequence that is about 80% to about 100% identical to SEQ ID NO: 4.

16 . The Gal-1/Gal-3 polynucleotide of claim 13 , wherein the alpha helix coil has a sequence that is about 80% to about 100% identical to SEQ ID NO: 5.

17 . A vector comprising:

the Gal-1/Gal-3 polynucleotide of claim 13 .

18 . A bacterial cell comprising:

the polynucleotide sequence of claim 13 .

19 . A method for reducing inflammation comprising: administering the Galectin-1/Galectin-3 (Gal-1/Gal-3) dimer of claim 1 or a pharmaceutical formulation comprising the Galectin-1/Galectin-3 (Gal-1/Gal-3) dimer of claim 1 to a subject in need thereof.

Assignments (2)
CONFIRMATORY LICENSE Recorded Dec 12, 2023
From: UNIVERSITY OF FLORIDA
To: NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT
Reel/Frame 065967/0438 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Nov 22, 2021
From: HUDALLA, GREGORY ALLAN; FETTIS, MARGARET MARY
To: UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INCORPORATED
Reel/Frame 058176/0623 →
Continuity (2)
Provisional Application 62811771 · Feb 28, 2019
Related Publication 20220098258A1 · Mar 31, 2022
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