IP Library Granted Patent US 11,839,596
Granted Patent B2
US 11,839,596 · App. 17/469,745 · Granted Dec 12, 2023

Treatment of vasculopathy with prostacyclin and mesenchymal stem cells

Inventors: Roger Jeffs (Chapel Hill, NC); Thomas Petersen (Durham, NC); Roger M. Ilagan (Burlington, NC); Michael Wade (Chapel Hill, NC)
Assignee: United Therapeutics Corporation
A61K31/192A61K31/557A61K35/28C12N5/0663C12N2501/00C12N2501/02
View Patent ↗
Loading inventors, assignments & file history…
Monitor This Case
Get email alerts when status or documents change.
Order Certified Copies
Most orders are placed with the USPTO same day — all within 24 business hours.
Order via The Patent Place →
Pre-filled with this patent's details
Quick Facts
Patent No.
US 11,839,596
App. No.
17/469,745
Granted
Dec 12, 2023
Kind
B2
Abstract

Provided are methods for treating or preventing vasculopathy in a subject in need thereof, comprising administering to the subject a prostacyclin and a mesenchymal stem cell (MSC) or a MSC-conditioned culture medium or administering to the subject a MSC or a MSC-conditioned culture medium that has treated with prostacyclin. Pharmaceutical compositions suitable for such treatments are also provided.

Claims (7)

1. A pharmaceutical composition comprising treprostinil or a pharmaceutically acceptable salt or ester thereof and a pharmaceutically effective amount of exosomes and a pharmaceutically acceptable carrier, wherein the exosomes are isolated from a mesenchymal stem cell culture comprising mesenchymal stem cells and treprostinil or a pharmaceutically acceptable salt or ester thereof, wherein the treprostinil or pharmaceutically acceptable salt or ester thereof is present in an amount sufficient to increase the amount of vascular endothelial growth factor contained in the mesenchymal stem cell culture and wherein the exosomes have increased VEGF-A gene transcript levels relative to exosomes obtained from a mesenchymal stem cell culture to which a prostacyclin was not added during culturing.

2. The pharmaceutical composition of claim 1 , wherein the amount of the treprostinil or pharmaceutically acceptable salt or ester thereof added to the culture medium is between about 200 μg/mL and about 300 μg/mL.

3. The pharmaceutical composition of claim 1 , wherein the mesenchymal stem cell is obtained from bone marrow.

4. The pharmaceutical composition of claim 1 , wherein the mesenchymal stem cell is a mesenchymal precursor cell.

5. The pharmaceutical composition of claim 1 , wherein the exosomes have at least about 4-fold increased VEGF-A gene transcript levels relative to exosomes obtained from a mesenchymal stem cell culture to which a prostacyclin was not added during culturing.

6. The pharmaceutical composition of claim 1 , wherein the exosomes have diameter from about 150 nm to about 200 nm.

7. The pharmaceutical composition of claim 1 , wherein about 60% of the exosomes have diameter of about 200 nm.

Continuity (4)
Division 16137629 · Sep 21, 2018
Division 14149929 · Jan 8, 2014
Provisional Application 61750458 · Jan 9, 2013
Related Publication 20220062210A1 · Mar 3, 2022
Cited By (1)
US 12,274,684