IP Library Granted Patent US 12,391,738
Granted Patent B2
US 12,391,738 · App. 17/895,638 · Granted Aug 19, 2025

Insulin-transferrin fusion protein and its prodrug, proinsulin-transferrin, for overcoming insulin resistance

Inventors: Wei-Chiang Shen (San Marino, CA); Yuqian Liu (Henan, CN); Hsuan-Yao Wang (Fullerton, CA)
Assignee: Livactus, Inc.
C07K14/62A61P3/00C07K14/79A61K38/00C07K2319/00
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Quick Facts
Patent No.
US 12,391,738
App. No.
17/895,638
Granted
Aug 19, 2025
Kind
B2
Abstract

A method of treating Type 2 diabetes (T2D) is provided. The method includes administering to a subject in need thereof an effective amount of a pharmaceutical composition that includes an insulin-transferrin fusion protein or its prodrug, proinsulin-transferrin fusion protein.

Claims (8)

1. A method of treating insulin resistance in a subject having insulin resistance comprising administering to the subject an effective amount of a pharmaceutical composition comprising a fusion protein encoded by a nucleic acid sequence comprising a pre-proinsulin nucleic acid sequence operably linked to a transferrin (Tf) sequence and a pharmaceutically acceptable carrier, thereby treating the insulin resistance.

2. The method of claim 1 , wherein the insulin resistance is associated with a disease selected from the group consisting of non-alcoholic fatty liver disease (NAFLD), nonalcoholic steatohepatitis (NASH) and Type 2 diabetes.

3. The method of claim 1 , wherein the subject's blood glucose level is at a level of a non-diabetic subject after treatment.

4. The method of claim 1 , wherein administration is in single-dosage form.

5. The method of claim 1 , wherein blood glucose levels are reduced within about 4-8 hours of administration.

6. The method of claim 1 , wherein the subject is a human.

7. The method of claim 1 , wherein the pharmaceutical composition is formulated for oral, parenteral, topical or rectal administration.

8. The method of claim 1 , wherein the pharmaceutically acceptable carrier is a liposome, a nanoparticle, a saline solution, water, a solvent, a buffer or another diluent.

Assignments (1)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Oct 14, 2022
From: SHEN, WEI-CHIANG; LIU, YUQIAN; WANG, HSUAN-YAO
To: LIVACTUS, INC.
Reel/Frame 061430/0705 →
Continuity (3)
Continuation 16630322
Provisional Application 62532822 · Jul 14, 2017
Related Publication 20220402993A1 · Dec 22, 2022
References Cited (12)
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Bailey, Clifford J., “Treating Insulin Resistance: Future Prospects,” [cited by applicant]
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Scarlett et al., “Insulin Treatment Reverses the Insulin Resistance of Type II Diabetes Mellitus,” [cited by applicant]
Wang et al., “Receptor-Mediated Activation of a Proinsulin-Transferrin Fusion Protein in Hepatoma Cells,” [cited by applicant]
Wang et al., “Proinsulin-Transferrin Fusion Protein as a Novel Long-Acting Insulin Analog for the Inhibition of Hepatic Glucose,” [cited by applicant]