IP Library › Granted Patent US 11,958,845
Granted Patent B2
US 11,958,845 · App. 17/952,546 · Granted Apr 16, 2024

Heterocyclic compound

Inventors: Masahiro Ito (Kanagawa, JP); Hideyuki Sugiyama (Kanagawa, JP); Takeshi Yamamoto (Kanagawa, JP); Keiko Kakegawa (Kanagawa, JP); Jinxing Li (Kanagawa, JP); Junsi Wang (Kanagawa, JP); Takahito Kasahara (Kanagawa, JP); Masato Yoshikawa (Kanagawa, JP)
Assignee: Takeda Pharmaceutical Company Limited
C07D413/14A61P25/28C07D413/10
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Quick Facts
Patent No.
US 11,958,845
App. No.
17/952,546
Granted
Apr 16, 2024
Kind
B2
Abstract

The present invention provides a heterocyclic compound having a HDAC6 inhibitory action, which is useful for the treatment of central nervous system diseases including neurodegenerative diseases, and the like, and a medicament comprising the compound. The present invention relates to a compound represented by the formula (I): wherein each symbol is as defined in the description, or a salt thereof.

Claims (4)

1. A method of inhibiting histone deacetylase 6 in a mammal, which comprises administering to the mammal an effective amount of a compound represented by formula (I) or a salt thereof:

wherein R 1 is an optionally substituted cyclic group, and R 2 is an optionally substituted cyclic group.

2. A method for treatment of Alzheimer's disease, progressive supranuclear palsy, frontotemporal dementia and parkinsonism linked to MAPT mutation (FTDP-17), frontotemporal dementia, Charcot-Marie-Tooth disease, peripheral neuropathy, amyotrophic lateral sclerosis (ALS) or cancer in a mammal, which comprises administering to the mammal an effective amount of a compound represented by formula (I) or a salt thereof:

wherein R 1 is an optionally substituted cyclic group, and R 2 is an optionally substituted cyclic group.

Priority Claims (1)
JP 2019-177815 · Sep 27, 2019 · national
Continuity (2)
Division 17030504 · Sep 24, 2020
Related Publication 20230183227A1 · Jun 15, 2023