IP Library › Granted Patent US 12,077,537
Granted Patent B2
US 12,077,537 · App. 18/110,126 · Granted Sep 3, 2024

Capsid inhibitors for the treatment of HIV

Inventors: Chienhung Chou (Dublin, CA); Scott E. Lazerwith (San Francisco, CA); John O. Link (San Francisco, CA); Scott D. Schroeder (Union City, CA); Winston C. Tse (Redwood City, CA); Jennifer R. Zhang (Union City, CA)
Assignee: Gilead Sciences, Inc.
C07D471/04A61K45/06C07D403/12C07D498/04C07D513/04C07D519/00
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Quick Facts
Patent No.
US 12,077,537
App. No.
18/110,126
Granted
Sep 3, 2024
Kind
B2
Abstract

The present disclosure relates generally to certain compounds, pharmaceutical compositions comprising said compounds, and methods of making and using said compounds and pharmaceutical compositions. The compounds and compositions disclosed herein may be used for the treatment or prevention of a Retroviridae viral infection, including an infection caused by the HIV virus.

Claims (10)

1. A compound that is selected from the group consisting of:

or a pharmaceutically acceptable salt thereof.

2. A compound that is selected from the group consisting of

or a pharmaceutically acceptable salt thereof.

3. A pharmaceutical composition comprising a compound of claim 1 , or a pharmaceutically acceptable salt thereof, and a pharmaceutically acceptable excipient or carrier.

4. A method of treating or preventing a human immunodeficiency virus (HIV) infection in a subject in need thereof, comprising administering to the subject a therapeutically effective amount of the compound of claim 1 , or a pharmaceutically acceptable salt thereof.

5. The method of claim 4 , further comprising administering a therapeutically effective amount of one or more additional therapeutic agents, or a pharmaceutically acceptable salt thereof.

6. A pharmaceutical composition comprising a compound of claim 2 , or a pharmaceutically acceptable salt thereof, and a pharmaceutically acceptable excipient or carrier.

7. A method of treating or preventing a human immunodeficiency virus (HIV) infection in a subject in need thereof, comprising administering to the subject a therapeutically effective amount of the compound of claim 2 , or a pharmaceutically acceptable salt thereof.

8. The method of claim 7 , further comprising administering a therapeutically effective amount of one or more additional therapeutic agents, or a pharmaceutically acceptable salt thereof.

Assignments (2)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jun 23, 2023
From: CHOU, CHIENHUNG; KATO, DARRYL; LAZERWITH, SCOTT E.; SCHROEDER, SCOTT D.; TSE, WINSTON C.; ZHANG, JENNIFER R.
To: GILEAD SCIENCES, INC.
Reel/Frame 064043/0077 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jun 23, 2023
From: LINK, JOHN O.
To: GILEAD SCIENCES, INC.
Reel/Frame 064043/0088 →
Continuity (3)
Continuation 17357376 · Jun 24, 2021
Provisional Application 63044086 · Jun 25, 2020
Related Publication 20230312567A1 · Oct 5, 2023
Cited By (3)
US 12,492,189 US 12,594,267 US 12,636,279