IP Library › Granted Patent US 12,377,098
Granted Patent B2
US 12,377,098 · App. 18/295,476 · Granted Aug 5, 2025

Compositions and methods for the treatment of alopecia

Inventor: Ofer A. Goren (Prague, CZ)
Assignee: FOLLEA INTERNATIONAL
A61K31/506A61K9/20A61K45/06A61P17/00
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Quick Facts
Patent No.
US 12,377,098
App. No.
18/295,476
Granted
Aug 5, 2025
Kind
B2
Abstract

Embodiments relate to compositions and methods for the treatment of hair loss, which can include treatment of alopecia, via an application of a composition including an alkalizing agent and/or a sulfotransferase enzyme. The composition can be formulated to be an orally administered composition. In some embodiments, the composition is used to increase the response of minoxidil.

Claims (28)

1. A method for improving, increasing, or enhancing hair re-growth of a subject suffering from alopecia, the method comprising:

orally administering a composition comprising an alkalizing agent and a sulfotransferase enzyme to a subject suffering from alopecia, thereby promoting sulfotransferase enzyme expression in an outer root sheath of a hair follicle of the subject.

2. The method of claim 1 ,

further comprising administering the composition further involves administering the composition topologically, via injection, or transdermally; and/or

administering the composition as a drug, a nutritional supplement, or a cosmetic.

3. The method of claim 1 , further comprising:

administering the composition before, during, and/or after administration of minoxidil.

4. The method of claim 1 ,

the composition further comprises minoxidil.

5. The method of claim 1 , wherein:

the alkalizing agent comprises one or more of a bicarbonate, citrate, a loop diuretic, MOPS, BES, TES, HEPES, DIPSO, TAPSO, Acetamidoglycine, POPSO, HEPPSO, HEPPS, Tricine, Tris (tromethamine), Glycinamide, Glycylglycine, Bicine, or TAPS.

6. The method of claim 1 , wherein:

the sulfotransferase enzyme comprises a human sulfotransferase enzyme and/or a non-human sulfotransferase enzyme.

7. The method of claim 1 , wherein:

the sulfotransferase enzyme comprises one or more of a carbohydrate sulfotransferase, a galactose-3-O-sulfotransferase, a heparan sulfate 2-O-sulfotransferase, a heparan sulfate 3-O-sulfotransferase, a heparan sulfate 6-O-sulfotransferase, a N-deacetylase/N-sulfotransferase, a tyrosylprotein sulfotransferase, an uronyl-2-sulfotransferase, an estrone sulfotransferase, a chondroitin 4-sulfotransferase, SULT1A1, SULT1A2, SULT1A3, SULT1A4, SULT1B1, SULT1C2, SULT1C3, SULT1C4, SULT1D1P, SULT1E1, SULT2A1, SULT2B1, SULT4A1, or SULT6B1.

8. The method of claim 1 , wherein:

the composition contains natural levels or extracts of minoxidil sulfotransferase enzymes, natural levels or extracts of phenol sulfotransferase enzymes, and/or natural levels of extracts sulfotransferase enzymes derived from Populus trichocarpa, Populus x canescens, Salix sp., Arabidopsis thaliana , silver poplar ( Populus alba ), Simon's poplar ( Populus simonii ), S. purpurea, P. tremuloides, I. polycarpa, P. nigra, Oryza sativa , Salicaceae family, Poplars ( Populus sp.), Idesia polycarpa , Japanese orange cherry, Potato ( Solanum tuberosum ), Cabbage ( Brassica rapa ), Populus trichocarpa (Black cottonwood), Salix Sp. (Willow tree), Cotton ( Gossypium ), Olea europaea L, Brassica napus, Apium graveolens, Brassica oleracea, Saccharina japonica, Solanum tuberosum , and/or Black cottonwood; and

the natural levels or extracts of minoxidil sulfotransferase enzymes, phenol sulfotransferase enzymes, and/or sulfotransferase enzymes are present in amounts ranging from 1%-100% by weight.

9. The method of claim 1 , wherein:

the sulfotransferase enzyme comprises OeST1.

10. The method of claim 1 , further comprising:

quantifying activity of SULT1A1 in dermal papillae cells and/or dermal sheath of the subject.

11. The method of claim 10 , further comprising:

determining a dosage and/or treatment regimen for the composition based on the quantitative measurement of activity of SULT1A1 in dermal papillae cells and/or dermal sheath of the subject.

12. A method for improving, increasing, or enhancing minoxidil response to a subject suffering from alopecia, the method comprising:

performing the method of claim 1 while the subject is undergoing minoxidil treatment for the alopecia.

13. A method for increasing sulfotransferase enzyme activity in a scalp and/or a liver of a subject suffering from alopecia, the method comprising:

orally administering a composition comprising an alkalizing agent and a sulfotransferase enzyme to a subject suffering from alopecia, thereby promoting sulfotransferase enzyme expression in an outer root sheath of a hair follicle of the subject.

Assignments (1)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Mar 7, 2025
From: GOREN, OFER A.
To: FOLLEA INTERNATIONAL
Reel/Frame 070436/0391 →
Continuity (4)
Provisional Application 63490939 · Mar 17, 2023
Provisional Application 63488045 · Mar 2, 2023
Provisional Application 63485333 · Feb 16, 2023
Related Publication 20240277709A1 · Aug 22, 2024
References Cited (9)
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Supikova, K.; Kosinova, A.; et al. “Sulfated phenolic acids in plants” Planta. May 13, 2022;255(6):124. (Year: 2022). [cited by examiner]
International Search Report and Written Opinion for PCT/US2023/017414 filed Apr. 4, 2023, dated Nov. 6, 2023. [cited by applicant]