IP Library › Granted Patent US 12,467,931
Granted Patent B2
US 12,467,931 · App. 18/354,151 · Granted Nov 11, 2025

Digital protein quantification

Inventors: Jeremy Agresti (Richmond, CA); Ronald Lebofsky (Kensington, CA)
Assignees: Bio-Rad Laboratories, Inc.; Bio-Rad Europe GmbH
G01N33/6878B01J19/0046C12Q1/6816C12Q1/6869C40B20/04C40B70/00
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Quick Facts
Patent No.
US 12,467,931
App. No.
18/354,151
Granted
Nov 11, 2025
Kind
B2
Abstract

Methods and compositions are described for single cell resolution, quantitative proteomic analysis using high throughput sequencing.

Claims (24)

1 . A method comprising:

incubating a plurality of permeabilized cells with a plurality of structurally distinct binding elements, each binding element having a specific binding affinity for a target epitope of a cellular protein, and wherein each binding element is conjugated to an epitope-specific oligonucleotide (ESO) comprising a barcode sequence specific to the target epitope, thereby binding the binding elements to their corresponding epitopes to form binder-epitope complexes;

washing away unbound binding elements;

isolating single cells of the plurality of permeabilized cells into a partition of a plurality of partitions;

providing to partitions of the plurality of partitions a plurality of partition-specific oligonucleotides (PSO) linked to a bead, each PSO comprising a partition-specific barcode sequence and a unique molecular identifier (UMI); and

hybridizing, in one or more partitions, a PSO with an ESO and extending the hybridized PSO with a polymerase, thereby generating a nucleic acid comprising an ESO, a partition-specific barcode sequence, and a UMI.

2 . The method of claim 1 , wherein each partition-specific oligonucleotide further comprises a primer binding sequence.

3 . The method of claim 1 , wherein each binding element is an antibody.

4 . The method of claim 1 , wherein each binding element is an aptamer.

5 . The method of claim 1 , wherein the plurality of structurally distinct binding elements comprises a library of at least 10, and no more than about 10,000, structurally distinct antibodies conjugated to the epitope-specific oligonucleotides.

6 . The method of claim 1 , further comprising discarding partitions that do not contain a single cell or contain multiple cells.

7 . The method of claim 1 , further comprising discarding partitions that do not contain a single partition-specific barcode sequence or contain multiple partition-specific barcode sequences.

8 . The method of claim 1 , wherein the partition-specific oligonucleotides are covalently linked to a bead with a cleavable linker.

9 . The method of claim 1 , further comprising lysing the cells after the isolating step.

10 . The method of claim 1 , wherein the plurality of partitions comprise a primer that binds to a primer binding sequence.

11 . The method of claim 10 , wherein the primer binding sequence is within the epitope-specific oligonucleotides.

12 . The method of claim 1 , wherein the epitope-specific oligonucleotide comprises a unique molecular identifier.

13 . The method of claim 1 , wherein each binding element is conjugated to a unique molecular identifier (UMI).

14 . The method of claim 1 , wherein each epitope-specific oligonucleotide further comprises a universal primer binding site.

15 . The method of claim 1 , further comprising cleaving the epitope-specific oligonucleotide from each binding element to yield a cleaved antibody oligonucleotide and cleaving the partition-specific oligonucleotide linked to the bead to yield a cleaved partition-specific oligonucleotide.

16 . The method of claim 15 , further comprising amplifying the cleaved antibody oligonucleotide using a universal primer and the cleaved partition-specific oligonucleotide.

17 . The method of claim 1 , wherein the plurality of partitions comprise wells, microwells or nanowells.

18 . The method of claim 1 , wherein the plurality of partitions comprise droplets.

19 . The method of claim 10 , wherein the primer binding sequence is within the partition-specific oligonucleotides.

Assignments (3)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jan 11, 2024
From: BIO-RAD INNOVATIONS
To: BIO-RAD EUROPE GMBH
Reel/Frame 066098/0679 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jan 11, 2024
From: AGRESTI, JEREMY
To: BIO-RAD LABORATORIES, INC.
Reel/Frame 066100/0116 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jan 11, 2024
From: LEBOFSKY, RONALD
To: BIO-RAD INNOVATIONS
Reel/Frame 066100/0367 →
Continuity (3)
Continuation 15393445 · Dec 29, 2016
Provisional Application 62273249 · Dec 30, 2015
Related Publication 20230417765A1 · Dec 28, 2023
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