IP Library › Granted Patent US 12,324,791
Granted Patent B2
US 12,324,791 · App. 18/518,127 · Granted Jun 10, 2025

Mirdametinib treatment

Inventors: Uchenna H. Iloeje (Stamford, CT); Abraham J. Langseth (Stamford, CT); Todd Webster Shearer (Stamford, CT)
Assignee: SPRINGWORKS THERAPEUTICS, INC.
A61K31/166A61K9/0053A61K31/216A61K45/06A61P25/00A61P35/00
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Quick Facts
Patent No.
US 12,324,791
App. No.
18/518,127
Filed
Nov 22, 2023
Granted
Jun 10, 2025
Kind
B2
Art Unit
1622
USPC
514/617
Abstract

The present disclosure relates to a method for treating certain types of tumors or cancers, such as plexiform neurofibromas (PN), plexiform neurofibromas associated with neurofibromatosis type 1 (NF1-PN), by orally administering an effective amount of mirdametinib to the patient, where an amount of mirdametinib is administered on the first day of treatment to provide (i) an AUC 0-tau less than 400 ng·h/mL, (ii) a C max no more than 40 ng/mL, or (iii) both.

Claims (2)

1. A method of treating a human patient 8 years or older who has neurofibromatosis type 1 (NF1) associated inoperable plexiform neurofibromas (PN) comprising orally administering an effective amount of mirdametinib to the patient, wherein an amount of mirdametinib is administered on the first day of treatment to provide (i) an AUC 0-tau less than 400 ng·h/mL, (ii) a C max no more than 40 ng/mL, or (iii) both, wherein, during treatment, the patient suffers from acneiform rash.

2. The method of claim 1 , wherein the patient suffers from pustular rash.

Assignments (1)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Nov 22, 2023
From: ILOEJE, UCHENNA H; LANGSETH, ABRAHAM J; SHEARER, TODD
To: SPRINGWORKS THERAPEUTICS, INC.
Reel/Frame 065650/0448 →
Continuity (5)
Continuation 18334518 · Jun 14, 2023
Continuation 18185148 · Mar 16, 2023
Provisional Application 63321036 · Mar 17, 2022
Provisional Application 63321046 · Mar 17, 2022
Related Publication 20240173274A1 · May 30, 2024
References Cited (13)
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“NF Consortium Protocol, NF Protocol 106,”, A Phase 2 Trial of the MEK Inhibitor PD-0325901 in Adolescents and Adults with NF1-Associated Morbid Plexiform Neurofibromas, 2018, 89 pages. [cited by applicant]
Cited By (1)
US 12,667,560