IP Library Granted Patent US 12,280,033
Granted Patent B2
US 12,280,033 · App. 18/763,671 · Granted Apr 22, 2025

Pharmaceutical combination for the treatment of a cancer

Inventors: Carles Domènech Garcia (Cerdanyola del Vallès, ES); José Alberto Alfón Coriat (Cerdanyola del Vallès, ES); Héctor Pérez Montoyo (Cerdanyola del Vallès, ES); Miguel Francisco Segura Ginard (Cerdanyola del Vallès, ES); Jose Miguel Lizcano De Vega (Cerdanyola del Vallès, ES)
Assignee: ABILITY PHARMACEUTICALS S.L.
A61K31/282A61K31/201A61K31/337A61K33/243A61K45/06A61P35/04
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Quick Facts
Patent No.
US 12,280,033
App. No.
18/763,671
Granted
Apr 22, 2025
Kind
B2
Abstract

A pharmaceutical combination comprising (A): a polyunsaturated fatty acid and (B): a chemotherapeutic agent compound for the simultaneous, separate or sequential use in the treatment of a cancer in a human patient.

Claims (24)

1. A pharmaceutical combination for the treatment of cancer comprising:

(i) a Compound (A) which comprises a polyunsaturated fatty acid of formula COOH—CHOH—(CH 2 ) 6 —(CH—CH—CH 2 ) 2 —(CH 2 ) 3 —CH 3 (ABTL0812), a pharmaceutically acceptable salt thereof, or a combination thereof

and

(ii) a Compound (B) which comprises at least one chemotherapeutic agent compound selected from the group consisting of a platinum-based agent, a nucleotide analog or precursor analog, an inhibitor of topoisomerase, or a combination thereof; and,

wherein the cancer is a tumor.

2. The pharmaceutical combination of claim 1 , wherein Compound (A) comprises a sodium salt of ABTL0812.

3. The pharmaceutical combination of claim 1 , wherein the pharmaceutical combination is a single composition comprising both Compound (A) and Compound (B).

4. The pharmaceutical combination of claim 1 , wherein the platinum-based agent is oxaliplatin.

5. The pharmaceutical combination of claim 1 , wherein the nucleotide analog or precursor analog is fluorouracil.

6. The pharmaceutical combination of claim 1 , wherein the inhibitor of topoisomerase is irinotecan.

7. The pharmaceutical combination of claim 1 , wherein the platinum-based agent is oxaliplatin; the nucleotide analog or precursor analog is fluorouracil; and the inhibitor of topoisomerase is irinotecan.

8. A pharmaceutical combination for the treatment of a tumor comprising (i) ABTL0812, a pharmaceutically acceptable salt thereof, or a combination thereof, and, (ii) irinotecan.

9. A method to treat a tumor in a subject in need thereof comprising administering a therapeutically effective amount of a pharmaceutical combination of claim 8 to the subject.

10. A pharmaceutical combination for the treatment of a tumor comprising (i) ABTL0812, a pharmaceutically acceptable salt thereof, or a combination thereof; and, (ii) fluorouracil.

11. A method to treat a tumor in a subject in need thereof comprising administering a therapeutically effective amount of a pharmaceutical combination of claim 10 to the subject.

12. A method to treat a cancer in a subject in need thereof comprising administering a therapeutically effective amount of a pharmaceutical combination of claim 1 to the subject; wherein the cancer is a tumor.

13. The method of claim 12 , wherein the tumor is selected from the group consisting of endometrial cancer, breast cancer, squamous cell cancer, lung cancer, endometrial cancer, cholangiocarcinoma, neuroblastoma, adenocarcinoma, pancreatic cancer, glioblastoma, and head and neck cancer.

14. The method of claim 12 , wherein Compound (A) is administered orally.

15. The method of claim 12 , wherein Compound (A) is administered as (i) a dose between 200 mg and 2,000 mg of Compound (A); or, (ii) a dose between 1,200 mg and 1,400 mg of Compound (A).

16. The method of claim 12 , wherein Compound (A) is administered daily.

17. The method of claim 12 , wherein Compound (B) is administrated intravenously.

18. The method of claim 17 , wherein Compound (B) is administered intravenously via infusion solution or via infusion suspension.

19. The method of claim 12 , wherein Compound (A) and Compound (B) are administered simultaneously, separately, or sequentially.

20. The method of claim 12 , wherein the administration of a pharmaceutically effective amount of the pharmaceutical combination to the subject reduces tumor size, reduces tumor size progression, stabilizes tumor size, stabilizes tumor size progression, reduces metastasis formation, increases survival rate, or a combination thereof.

Assignments (2)
CHANGE OF NAME Recorded Mar 21, 2025
From: ABILITY PHARMACEUTICALS S.L.
To: ABILITY PHARMACEUTICALS SA
Reel/Frame 070586/0936 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jul 10, 2024
From: DOMÈNECH GARCIA, CARLES; ALFÓN CORIAT, JOSÉ ALBERTO; PÉREZ MONTOYO, HÉCTOR; SEGURA GINARD, MIGUEL FRANCISCO; LIZCANO DE VEGA, JOSE MIGUEL
To: ABILITY PHARMACEUTICALS S.L.
Reel/Frame 067952/0045 →
Priority Claims (1)
EP 17382282 · May 16, 2017 · regional
Continuity (3)
Continuation 17581587 · Jan 21, 2022
Continuation 16614084
Related Publication 20240350449A1 · Oct 24, 2024
References Cited (18)
US 8735436B2 · Hovland et al. · 2014 [cited by applicant]
US 9050308B2 · Maines et al. · 2015 [cited by applicant]
US 11260042B2 · Domènech García et al. · 2022 [cited by examiner]
US 12053449B2 · Domènech García et al. · 2024 [cited by examiner]
US 20040053882A1 · Smith et al. · 2004 [cited by applicant]
US 20060058311A1 · Munzert et al. · 2006 [cited by applicant]
US 20140271562A1 · Garcia-Rodenas et al. · 2014 [cited by applicant]
EP 2409963B1 · 2017 [cited by applicant]
RU 2284818C2 · 2004 [cited by applicant]
WO WO2018210830A1 · 2018 [cited by applicant]
AbilityPharmaceuticalsAnnouncesFDA-Orphan Drug Designationfor ABTLO0812inPancreaticCancer, Dec. 14, 2016, accessedat https/avwow.abillitvpharma.com/on/mainimenu/media-centerpresse-reloase/abihity˜pharmaceuticals-announc… [cited by examiner]
AbilityPharma, “Ability Pharmaceuticals Announces FDA-Orphan Drug Designation for ABTL0812 in Pancreatic Cancer”, Dec. 14, 2016, accessed at https://www.abilitypharma.com/en/main-menu/media-center/press-release/ability-… [cited by applicant]
AbilityPharma, “Ability Pharmaceuticals Initiates Phase 2 Combination Trial with ABTL0812 as First Line Therapy in Patients with Endometrial or Squamous Lung Cancer Patients”, Nov. 22, 2016, accessed at https://www.abil… [cited by applicant]
Alfon, J., et al., “Effect of ABTL0812, a safe dual inhibitor of mTORC1/C2 and dihydrofolate reductase, on gemcitabine and docetaxel cytotoxicity in pancreatic and lung cancer cells,” Journal of Clinical 31:15, American… [cited by applicant]
Colas, E., et al., “The first-in-class anti-cancer agent ABTL0812 is effective in preclinical models of human endometrial cancer,” Journal of Clinical Oncology 35(15):e17070, American Society for Clinical Cancer Researc… [cited by applicant]
Erazo, T., et al., “The New Antitumor Drug ABTL0812 Inhibits the Akt/mTORCI Axis by Upregulating Tribbles-3 Pseudokinase,” Clin Cancer Res. 22(10):2508-2519, American Association for Cancer Research, United States (May … [cited by applicant]
International Search Report and Written Opinion for International Application No. PCT/EP2018/062554, European Patent Office, Netherlands, mailed on Aug. 3, 2018, 10 pages. [cited by applicant]
Google Patents, English-language Machine Translation of Russian Patent RU-2284818-C2, performed on Mar. 4, 2024, 9 pages. [cited by applicant]