IP Library Granted Patent US 12,178,801
Granted Patent B1
US 12,178,801 · App. 18/818,317 · Granted Dec 31, 2024

Stable psilocin salts, esters and conjugates and uses thereof

Inventors: Yousry Sayed (Wilmington, NC); Frederick Sancilio (Stuart, FL); Shaileshkumar Ramanlal Desai (Wilmington, NC); Autumn Beauchamp (Wilmington, NC)
Assignee: Lobe Sciences Ltd.
A61K31/4045A61K47/542
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Quick Facts
Patent No.
US 12,178,801
App. No.
18/818,317
Granted
Dec 31, 2024
Kind
B1
Abstract

Pharmaceutically acceptable salts, esters and conjugates of psilocin and compositions and methods for their production and use in treating diseases or conditions treatable with psilocin or psilocybin are provided.

Claims (8)

1. A composition comprising a psilocin mucate salt or conjugate.

2. The composition of claim 1 which exhibits improved stability as compared to psilocin.

3. A pharmaceutical composition comprising the composition of claim 1 and one or more pharmaceutically acceptable excipients.

4. A method for producing the composition of claim 1 comprising mixing psilocin with galactaric acid (mucic acid).

5. A method for treating a disease or condition in a subject treatable with psilocin or psilocybin, said method comprising administering to the subject the composition of claim 1 .

6. The method of claim 5 wherein the disease or condition is a neurological injury, neurodegenerative disease, neurological disorder, neurodevelopmental disorder, inflammatory condition, chronic pain, or a psychological condition.

7. The method of claim 5 wherein the disease or condition is chronic cluster headaches.

8. A method of reducing adverse effects of psilocybin or psilocin administration in a subject, said method comprising administering to the subject the composition of claim 1 .

Assignments (2)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jul 17, 2025
From: LOBE SCIENCES LTD.
To: CYNAPTEC PHARMACEUTICALS, INC.
Reel/Frame 071744/0638 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Sep 4, 2024
From: SAYED, YOUSRY; SANCILIO, FREDERICK; DESAI, SHAILESHKUMAR RAMANLAL; BEAUCHAMP, AUTUMN
To: LOBE SCIENCES LTD.
Reel/Frame 068485/0008 →
Continuity (2)
Continuation In Part PCTUS2023027500 · Jul 12, 2023
Provisional Application 63388414 · Jul 12, 2022
Cited By (1)
US 12,344,583